Search Results
38286 articles found
REVIEW
|
doi:10.20944/preprints202405.0059.v1
Subject:
Medicine And Pharmacology,
Dermatology
Keywords:
atopic dermatitis; calcineurin; NFAT; tacrolimus; pimecrolimus; cyclosporine
Online: 1 May 2024 (07:49:16 CEST)
ARTICLE
|
doi:10.20944/preprints202406.0034.v1
Subject:
Biology And Life Sciences,
Neuroscience And Neurology
Keywords:
voltage-gated sodium channels; fibroblast growth factors; split luciferase assay; kinase inhibitors
Online: 3 June 2024 (08:07:35 CEST)
REVIEW
|
doi:10.20944/preprints202404.0944.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Immune checkpoint inhibitor; ipilimumab; pembrolizumab
Online: 16 April 2024 (03:30:17 CEST)
REVIEW
|
doi:10.20944/preprints202405.0668.v3
Subject:
Biology And Life Sciences,
Neuroscience And Neurology
Keywords:
epilepsy; neuroinflammation; NLRP3 inflammasome; epileptogenesis; antiseizure medication; interleukin-1b; caspase-1; ASC
Online: 31 May 2024 (15:29:49 CEST)
ARTICLE
|
doi:10.20944/preprints201609.0074.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
hepatocellular carcinoma; hepatitis B virus X protein; Notch1 pathway; ERK; AKT
Online: 21 September 2016 (09:49:13 CEST)
REVIEW
|
doi:10.20944/preprints202012.0675.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Breast cancer; Estrogen Receptor; PI3K-AKT-mTOR; anti-estrogen resistance
Online: 28 December 2020 (09:22:17 CET)
REVIEW
|
doi:10.20944/preprints202309.0682.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
Akt; cancer; metastasis; HNSCC; EMT; cytoskeletal remodelling
Online: 12 September 2023 (08:33:01 CEST)
REVIEW
|
doi:10.20944/preprints202307.1695.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
hepatocellular carcinoma; EGFR/PI3K/AKT/mTOR signaling; animal models; Targeted Therapy
Online: 26 July 2023 (10:07:16 CEST)
REVIEW
|
doi:10.20944/preprints202402.0872.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Immunotherapy; Immune checkpoint inhibitors; Rechallenge therapy; Resistance; NSCLC
Online: 16 February 2024 (11:34:11 CET)
ARTICLE
|
doi:10.20944/preprints202106.0443.v1
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
miR-378d; ESCC; AKT; RhoA; polyploidization
Online: 16 June 2021 (12:07:30 CEST)
REVIEW
|
doi:10.20944/preprints202406.0880.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Dendritic cells; DC based cancer vaccine; Immune checkpoint inhibitors; Cancer Therapy; Combinatorial therapy
Online: 13 June 2024 (11:51:42 CEST)
REVIEW
|
doi:10.20944/preprints202408.0744.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
Peripheral T-cell lymphoma; Histone deacetylase (HDAC); HDAC inhibitor (HDACi); targeted therapy; epigenetic; DNA mutation; TET2; DNMT3A
Online: 12 August 2024 (05:07:04 CEST)
ARTICLE
|
doi:10.20944/preprints202004.0312.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
chalocomoracin; proliferative vitreoretinopathy; vitreous; Akt; p53; migration; proliferation; contraction
Online: 19 April 2020 (02:18:01 CEST)
ARTICLE
|
doi:10.20944/preprints202403.0717.v1
Subject:
Biology And Life Sciences,
Animal Science, Veterinary Science And Zoology
Keywords:
Lumpy skin disease; DNA polymerase; potential inhibitors; phytocompounds; antiviral drug compounds; molecular docking
Online: 13 March 2024 (07:58:39 CET)
REVIEW
|
doi:10.20944/preprints202205.0290.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
Cholesterol; PCSK9 inhibitors; HMG-CoA; LDL receptor; statins
Online: 23 May 2022 (10:01:24 CEST)
ARTICLE
|
doi:10.20944/preprints202107.0228.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Myopia; monocular form deprivation (MFD); inflammation; Fallopia Japonica (FJ); Prunella Vulgaris (PV)
Online: 9 July 2021 (15:21:52 CEST)
REVIEW
|
doi:10.20944/preprints202404.0091.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
menin; menin inhibitors; leukemia; KMT2A; NPM1
Online: 2 April 2024 (02:51:43 CEST)
ARTICLE
|
doi:10.20944/preprints202408.2012.v1
Subject:
Biology And Life Sciences,
Other
Keywords:
Herbacetin; (-)-Epicatechin; KATII inhibition; molecular docking; Molecular dynamic
Online: 28 August 2024 (09:37:19 CEST)
ARTICLE
|
doi:10.20944/preprints202404.1491.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
HIV-2; integrase strand transfer inhibitor (INSTIs); HIV; integrase; Lenacapavir; SARs-CoV-2
Online: 23 April 2024 (05:06:50 CEST)
ARTICLE
|
doi:10.20944/preprints202407.0477.v1
Subject:
Medicine And Pharmacology,
Epidemiology And Infectious Diseases
Keywords:
DENV3; ZIKV; molecular docking; MD simulations; MM/GBSA; compound library; NS5; lycorine
Online: 5 July 2024 (12:04:10 CEST)
ARTICLE
|
doi:10.20944/preprints202407.1450.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Bladder cancer; STAT3 inhibitor; Apoptosis; Preclinical; 3D models
Online: 17 July 2024 (14:18:54 CEST)
ARTICLE
|
doi:10.20944/preprints202409.0421.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Helicobacter pylori; antimicrobial resistance; narrow-spectrum antibiotic; antibacterial target; response regulator; HsrA; Campylobacter jejuni
Online: 5 September 2024 (10:22:25 CEST)
REVIEW
|
doi:10.20944/preprints202402.1049.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
malignant pleural mesothelioma; immune checkpoint inhibitor; orphan drug; good clinical practice; Pharmaceuticals and Medical Devices Agency
Online: 20 February 2024 (04:03:22 CET)
ARTICLE
|
doi:10.20944/preprints202406.2011.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
machine learning; prediction methods; cancer; ic50; r programming
Online: 29 June 2024 (05:59:44 CEST)
ARTICLE
|
doi:10.20944/preprints202402.1740.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Rheumatoid Arthritis, Anti-TNF, NRF2, Reverse Signaling, Biotherapy, Monoclonal Antibodies, Monocytes, Prediction.
Online: 29 February 2024 (14:46:26 CET)
ARTICLE
|
doi:10.20944/preprints202403.1880.v1
Subject:
Public Health And Healthcare,
Other
Keywords:
Anti-interferon-γ autoantibodies; herpes zoster; monocyte chemoattractant protein-1; IFN-γ inducible protein-10; Janus kinas inhibitors; rheumatoid arthritis.
Online: 1 April 2024 (10:20:44 CEST)
ARTICLE
|
doi:10.20944/preprints202405.1741.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
Alzheimer’ s disease; vascular complications; monoclonal antibody therapy; Aducanumab; Lecanemab; epoxide of polyunsaturated fatty acid; soluble epoxide hydrolase inhibitor EC5026; EP4 inhibitor; monocyte/macrophage; amyloid-beta degradation
Online: 27 May 2024 (13:00:54 CEST)
BRIEF REPORT
|
doi:10.20944/preprints202403.0928.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
systemic sclerosis; pulmonary hypertension; Phosphodiesterase-5 inhibitors; endothelin receptor antagonist
Online: 15 March 2024 (13:15:50 CET)
ARTICLE
|
doi:10.20944/preprints201909.0189.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
miR-139-5p; SLC7A11; proliferation; migration; pancreatic cancer (PANC)
Online: 17 September 2019 (12:42:14 CEST)
ARTICLE
|
doi:10.20944/preprints201804.0082.v2
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Resveratrol; TRAIL; apoptosis; lung cancer cells; NF-κB; Cytochrome c
Online: 13 August 2018 (06:18:03 CEST)
ARTICLE
|
doi:10.20944/preprints201808.0043.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
cryptotanshinone; NSCLC; cell cycle arrest; apoptosis; PI3K/Akt/GSK3β
Online: 2 August 2018 (09:05:32 CEST)
ARTICLE
|
doi:10.20944/preprints201807.0297.v1
Subject:
Biology And Life Sciences,
Food Science And Technology
Keywords:
24-methylenecycloartanyl ferulate, angiogenesis, PPAR-γ2, PPRE, Akt/mTOR, HoxA7, VEGF, LIF, HUVEC
Online: 17 July 2018 (09:10:14 CEST)
ARTICLE
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
Metformin; cerebralischemia-reperfusion; inflammation; PI3K/Akt.
Online: 12 March 2021 (08:43:06 CET)
REVIEW
|
doi:10.20944/preprints202401.0310.v1
Subject:
Medicine And Pharmacology,
Dentistry And Oral Surgery
Keywords:
inflammation; inflammasome; inhibitors of the inflammasome; nanomaterials; functionalized biomaterials; periodontitis; general pathology
Online: 4 January 2024 (09:25:17 CET)
REVIEW
|
doi:10.20944/preprints202306.0441.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
anti-lipoxygenase peptide; bioactivity; enzymatic hydrolysis; food peptide; food protein; inflammation; lipoxidase; lipoxygenase inhibitory activity.
Online: 6 June 2023 (10:11:09 CEST)
REVIEW
|
doi:10.20944/preprints202405.0573.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
Proton Pump Inhibitors (PPIs); Vonoprazan (VPZ); Intravenous infusion; Oral therapy; Bleeding peptic ulcers; Endoscopic therapy
Online: 9 May 2024 (09:15:54 CEST)
ARTICLE
|
doi:10.20944/preprints202405.1890.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Parecoxib; 5-fluorouracil; Colorectal cancer; Metastasis; Reactive oxygen species; PI3K/Akt pathway
Online: 28 May 2024 (17:00:53 CEST)
ARTICLE
|
doi:10.20944/preprints201609.0123.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
carbonic anhydrase; acetylcholinesterase; β-Lactam; 2-Azetidinone; enzyme inhibition; enzyme purification
Online: 30 September 2016 (05:38:45 CEST)
ARTICLE
|
doi:10.20944/preprints202305.1949.v2
Subject:
Biology And Life Sciences,
Toxicology
Keywords:
Methamphetamine; BDNF; CREB; Akt-1; GSK3; Amygdala
Online: 20 September 2023 (03:22:53 CEST)
ARTICLE
|
doi:10.20944/preprints202008.0112.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
AKT/PI3K signaling pathway; apoptosis; human hepatocarcinoma HepG2 cells; migration activity; proliferation; oxidative stress; ROS level; uvaol
Online: 5 August 2020 (05:58:26 CEST)
ARTICLE
|
doi:10.20944/preprints202405.0035.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Mycobacterial Polyketide Synthase; QSAR; Multiple Linear Regression; Docking; Molecular Dynamics Simulations
Online: 1 May 2024 (16:46:55 CEST)
ARTICLE
|
doi:10.20944/preprints202304.0565.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Chrysomycin A; Xenograft mouse model; Glioblastoma; Apoptosis
Online: 19 April 2023 (08:00:29 CEST)
ARTICLE
|
doi:10.20944/preprints202305.0844.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Peptidomimetic; VEGFR2; Angiogenesis; Tumor suppression; PI3K/Akt/mTOR signaling pathway; PLCγ/ERK signaling pathway
Online: 11 May 2023 (10:57:38 CEST)
ARTICLE
|
doi:10.20944/preprints202404.1152.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Tuberculosis; nitrobenzamides; DprE; mycobacteria
Online: 17 April 2024 (11:50:50 CEST)
REVIEW
|
doi:10.20944/preprints202204.0202.v1
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
Metabolic syndrome; SGLT2 inhibitors; Dapagliflozin; Empagliflozin; Canagliflozin; Translational modeling
Online: 21 April 2022 (10:12:04 CEST)
REVIEW
|
doi:10.20944/preprints202012.0167.v2
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Matrix metalloproteinase; MMPs; protease; TIMPs; exosite; small molecule inhibitors; monoclonal antibodies; proteomics; N-terminomics; TAILS
Online: 24 March 2021 (16:23:28 CET)
ARTICLE
|
doi:10.20944/preprints202407.1916.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
cardiovascular disease; hepatic fibrosis; metabolic dysfunction-associated steatotic liver disease; sodium-glucose cotransporter 2 inhibitors; serum lipids
Online: 24 July 2024 (08:27:35 CEST)
REVIEW
|
doi:10.20944/preprints202401.0803.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
CYP enzymes; CYP3A4; flavonoid; inhibition; natural products
Online: 10 January 2024 (10:24:39 CET)
ARTICLE
|
doi:10.20944/preprints202307.0031.v1
Subject:
Chemistry And Materials Science,
Applied Chemistry
Keywords:
Ionic Liquids; Corrosion Inhibitors; Bio-based
Online: 4 July 2023 (02:23:59 CEST)
ARTICLE
|
doi:10.20944/preprints201710.0143.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
cheminformatics; docking simulation; drug repositioning; thiopurine; tyrosinase
Online: 22 October 2017 (14:03:13 CEST)
ARTICLE
|
doi:10.20944/preprints202406.0032.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
HIV-1; reverse transcriptase; polymerase; ribonuclease H; inhibitor; benzisothiazolone
Online: 3 June 2024 (07:56:06 CEST)
ARTICLE
|
doi:10.20944/preprints202308.0641.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
licochalcone H (LCH); oxaliplatin; colorectal cancer; EGFR; AKT; apoptosis
Online: 9 August 2023 (03:01:44 CEST)
ARTICLE
|
doi:10.20944/preprints201901.0018.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
pyruvate kinase M2; prostate cancer; cancer metabolism; mTOR; autophagy
Online: 3 January 2019 (12:32:52 CET)
ARTICLE
|
doi:10.20944/preprints201705.0218.v1
Subject:
Chemistry And Materials Science,
Food Chemistry
Keywords:
anticancer activity; apoptosis; oleanolic acid; cell cycle arrest; mapk signaling
Online: 31 May 2017 (11:28:30 CEST)
ARTICLE
|
doi:10.20944/preprints201910.0154.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
papillary thyroid cancer; germline mutations; whole genome sequencing; predisposition markers; pathway analysis
Online: 13 October 2019 (17:07:34 CEST)
ARTICLE
|
doi:10.20944/preprints202208.0103.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Resveratrol; antioxidant metabolism; scavengome; biomimetic oxidation; bioactivity-guided isolation; NMR spectroscopy; xanthine oxidase
Online: 4 August 2022 (05:33:52 CEST)
ARTICLE
|
doi:10.20944/preprints202408.0754.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
Zika Infection; Extracellular; Vesicles; Proteome; Metabolome; Network
Online: 12 August 2024 (04:52:50 CEST)
ARTICLE
|
doi:10.20944/preprints202106.0169.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
melanoma initiating cells; CD133; drug resistance; apoptosis; caspase activation; CRISPR-Cas9 knockout; AKT; BAD; BCL-2 family
Online: 7 June 2021 (12:11:10 CEST)
REVIEW
|
doi:10.20944/preprints202012.0419.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
immune checkpoint; lymphoid neoplasms; programmed death 1; cytotoxic T-lymphocyte antigen 4; monoclonal antibodies; combination therapies
Online: 17 December 2020 (08:10:05 CET)
ARTICLE
|
doi:10.20944/preprints202310.1571.v2
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Transketolase; malonylation; acetylation; sirtuin 5; oxythiamine; metformin; amprolium; thiamine; posttranslational modifications
Online: 10 November 2023 (12:03:31 CET)
REVIEW
|
doi:10.20944/preprints202406.0356.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
liver transplantation; hepatocellular carcinoma; Immune checkpoint inhibitors; allograft rejection
Online: 6 June 2024 (07:45:00 CEST)
ARTICLE
|
doi:10.20944/preprints201901.0250.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
drug delivery system, muscle atrophy, nanoparticle, prostaglandin E1, sciatic nerve injury
Online: 24 January 2019 (08:51:02 CET)
REVIEW
|
doi:10.20944/preprints202404.0176.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
histone deacetylase inhibitors; radiosensitisation; heterochromatin; double strand break; DNA repair
Online: 2 April 2024 (10:09:33 CEST)
REVIEW
|
doi:10.20944/preprints202308.1413.v1
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
diabetes; cardiovascular; renal; SGLT1; SGLT2; therapy.
Online: 22 August 2023 (07:45:50 CEST)
REVIEW
|
doi:10.20944/preprints202307.1892.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Oncolytic virus; immune checkpoint inhibitors; immunotherapy
Online: 28 July 2023 (10:58:30 CEST)
ARTICLE
|
doi:10.20944/preprints202012.0383.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
meprin α; meprin β; zinc metalloproteinase; medicinal chemistry; probe development
Online: 15 December 2020 (12:56:31 CET)
ARTICLE
|
doi:10.20944/preprints202012.0354.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
meprin α; meprin β; zinc metalloproteinase; uHTS
Online: 14 December 2020 (16:36:57 CET)
HYPOTHESIS
|
doi:10.20944/preprints202004.0151.v2
Online: 22 April 2020 (09:46:54 CEST)
ARTICLE
|
doi:10.20944/preprints202408.1642.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
allogeneic hematopoietic stem cell transplantation; chronic myeloid leukaemia; tyrosine kinase inhibitors; imatinib; dasatinib; nilotinib
Online: 22 August 2024 (16:30:22 CEST)
ARTICLE
|
doi:10.20944/preprints202310.1011.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Cucumis sativus; endothelial dysfunction; hypertension; pAkt, angiotensin-II, mice
Online: 17 October 2023 (04:50:09 CEST)
REVIEW
|
doi:10.20944/preprints202311.0295.v1
Subject:
Medicine And Pharmacology,
Cardiac And Cardiovascular Systems
Keywords:
Atrial fibrillation, SGLT2 inhibitors, cardiovascular outcomes, hemodynamic effects, AF risk reduction
Online: 6 November 2023 (08:13:49 CET)
ARTICLE
|
doi:10.20944/preprints202404.0785.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
enteroviruses, coxsackievirus, leucoverdazyls, antioxidant, antiviral, 2C protein
Online: 11 April 2024 (09:22:02 CEST)
REVIEW
|
doi:10.20944/preprints202401.1697.v1
Subject:
Medicine And Pharmacology,
Cardiac And Cardiovascular Systems
Keywords:
DOAC; FXIa; mAbs; ASO; drug-drug interactions
Online: 23 January 2024 (12:31:04 CET)
REVIEW
|
doi:10.20944/preprints202305.1761.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
checkpoint inhibitors; colitis; immune-related adverse events; enterocolitis; diarrhea
Online: 25 May 2023 (08:03:37 CEST)
ARTICLE
|
doi:10.20944/preprints202302.0423.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
B-cell; autoimmune disease; drug repurposing
Online: 24 February 2023 (09:11:37 CET)
REVIEW
|
doi:10.20944/preprints202402.1535.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
DNA polymerase I; Polymerase θ ; reverse transcriptase; homologous recombination; antibiotics; apicoplast
Online: 27 February 2024 (12:29:29 CET)
REVIEW
|
doi:10.20944/preprints202304.0516.v1
Subject:
Medicine And Pharmacology,
Internal Medicine
Keywords:
SGLT-2 Inhibitors; Inflammasome; NLRP3; reno-protective effects; Cardio-protective effects; neuro-protective effects.
Online: 18 April 2023 (10:33:39 CEST)
ARTICLE
|
doi:10.20944/preprints202211.0356.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Focal adhesion kinase; 3D-QSAR; Molecular Dynamics; MM-PB/GBSA; Free energy perturbation
Online: 18 November 2022 (10:13:00 CET)
ARTICLE
|
doi:10.20944/preprints202108.0001.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Antitumoral drug; Choline kinase inhibition; Choline uptake
Online: 2 August 2021 (08:42:22 CEST)
ARTICLE
|
doi:10.20944/preprints202001.0255.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
Cordycepin; Cisplatin-resistance; Resensitization; MDR1; Ets-1; AKT
Online: 22 January 2020 (09:18:20 CET)
ARTICLE
|
doi:10.20944/preprints202408.1759.v1
Subject:
Biology And Life Sciences,
Neuroscience And Neurology
Keywords:
HIV; ferritin heavy-chain; ferritin light-chain; ferroptosis; lipid peroxidation; iron; oxidative stress; neurocognitive impairment; neurocognitive domains
Online: 24 August 2024 (00:22:41 CEST)
ARTICLE
|
doi:10.20944/preprints202312.1461.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
indirect comparison; Shiny method; reconstructed individual patient data; disease free survival; renal cell carcinoma; adjuvant setting
Online: 20 December 2023 (09:30:07 CET)
ARTICLE
|
doi:10.20944/preprints201703.0116.v1
Subject:
Biology And Life Sciences,
Animal Science, Veterinary Science And Zoology
Keywords:
In vivo; Alpha-glucosidase; Alpha-amylase; hyperglycemia
Online: 16 March 2017 (09:35:36 CET)
ARTICLE
|
doi:10.20944/preprints201909.0091.v1
Subject:
Medicine And Pharmacology,
Dermatology
Keywords:
fisetin; psoriasis; normal human epidermal keratinocyte; cell signaling; cell differentiation; proliferation; inflammatory cytokine; PBMC; CD4+ T lymphocyte; 3D psoriasis-like skin disease model
Online: 9 September 2019 (07:48:26 CEST)
ARTICLE
|
doi:10.20944/preprints202408.1282.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Cataract; CRYGD; Molecular docking; Molecular dynamics; Crystallin; Protein aggregation
Online: 19 August 2024 (09:15:05 CEST)
ARTICLE
|
doi:10.20944/preprints202004.0240.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
COVID19; 2019-nCov, 3CLpro inhbitors
Online: 15 April 2020 (10:00:52 CEST)
ARTICLE
|
doi:10.20944/preprints202002.0047.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
2019-nCoV; therapeutic strategies; drug; ACE2
Online: 4 February 2020 (10:59:25 CET)
REVIEW
|
doi:10.20944/preprints201909.0140.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
hepatocellular carcinoma; immune checkpoint inhibitors; HCC; pembrolizumab; nivolumab; immune microenvironment; targeted therapies
Online: 14 September 2019 (18:37:29 CEST)
REVIEW
|
doi:10.20944/preprints201805.0145.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
carbonic anhydrase, enzyme inhibition, metalloenzymes, amino acid, glaucoma, tumors
Online: 9 May 2018 (13:55:15 CEST)
ARTICLE
|
doi:10.20944/preprints202311.0483.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
MRONJ; CDK4/6 inhibitors; metastatic breast cancer; oral epidemiology
Online: 8 November 2023 (08:42:55 CET)
ARTICLE
|
doi:10.20944/preprints202307.2034.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Bcl-2; Anti-apoptotic protein; Indole; Cancer drug discovery
Online: 28 July 2023 (14:36:37 CEST)
ARTICLE
|
doi:10.20944/preprints202107.0270.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
drug design; falcipain; malaria; peptidomimetics; Plasmodium falciparum; virtual screening; pharmacophore.
Online: 12 July 2021 (14:48:13 CEST)
REVIEW
|
doi:10.20944/preprints202106.0158.v1
Online: 7 June 2021 (09:29:06 CEST)
ARTICLE
|
doi:10.20944/preprints201811.0330.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
hyperpigmentation; tyrosinase inhibitors; 3-(2,4-dihydroxyphenyl)propionic acid; structure-activity relationship study; B16-F10 cellular melanogenesis inhibition
Online: 14 November 2018 (09:59:45 CET)
ARTICLE
|
doi:10.20944/preprints201801.0213.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
bichalcones; sirtuin inhibitors; virtual screening
Online: 23 January 2018 (09:12:43 CET)
ARTICLE
|
doi:10.20944/preprints202005.0445.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
oral cancer; cancer-associated fibroblasts; metastasis; cell migration; cell invasion; Akt; EGFR
Online: 27 May 2020 (08:25:20 CEST)
ARTICLE
|
doi:10.20944/preprints201706.0120.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
sinulariolide; human bladder cancer; migration; invasion; PI3K/AKT/mTOR signaling pathway
Online: 27 June 2017 (06:23:44 CEST)
ARTICLE
|
doi:10.20944/preprints202307.1251.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
ascorbic acid; pharmacologic ascorbate; pancreatic cancer; epigenetics; DNA methyltransferase (DNMT); ten-eleven translocation (TET) methylcytosine dioxygenase
Online: 18 July 2023 (13:51:14 CEST)
ARTICLE
|
doi:10.20944/preprints202301.0129.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
chondrogenesis; cartilage; col11a1; collagen α1(XI), AKT; GSK3b; Wnt; ATDC5
Online: 7 January 2023 (13:00:05 CET)
REVIEW
|
doi:10.20944/preprints202405.0992.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
proteases; viruses; respiratory proteases; protease inhibitors; SARS-CoV-2
Online: 15 May 2024 (10:29:30 CEST)