Search Results
31971 articles found
ARTICLE
|
doi:10.20944/preprints201910.0072.v1
Subject:
Chemistry And Materials Science,
Materials Science And Technology
Keywords:
Faraday rotation; Thin films; Magneto-optics; Organic material; Tolane derivatives
Online: 7 October 2019 (12:26:26 CEST)
ARTICLE
|
doi:10.20944/preprints202403.1557.v1
Subject:
Chemistry And Materials Science,
Polymers And Plastics
Keywords:
biodegradable polymers; antibacterial polymers; chitosan Schiff base; κ-carrageenan blend; grafted copolymer
Online: 26 March 2024 (11:30:13 CET)
ARTICLE
|
doi:10.20944/preprints202403.0479.v1
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
quinone; quinone imine; hydrogen bonding; X-ray crystallography; NMR titration; redox.
Online: 8 March 2024 (10:33:48 CET)
ARTICLE
|
doi:10.20944/preprints202403.0382.v1
Subject:
Chemistry And Materials Science,
Materials Science And Technology
Keywords:
donor-acceptor derivatives; blue organic light emitting diode; high efficiency; blue emission; thermal analysis
Online: 7 March 2024 (09:34:59 CET)
ARTICLE
|
doi:10.20944/preprints201605.0002.v1
Online: 11 May 2016 (07:42:45 CEST)
ARTICLE
|
doi:10.20944/preprints202402.0887.v1
Subject:
Chemistry And Materials Science,
Materials Science And Technology
Keywords:
Calixarene; Dihomooxacalixarene; Hexahomotrioxacalixarene; Pseudopolymorphism; X-ray diffraction
Online: 16 February 2024 (06:58:09 CET)
ARTICLE
|
doi:10.20944/preprints201703.0053.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
1,3,4-Thiadiazole; 1,2,4-Triazole; synthesis; MTT assay; Cytotoxicity of Schiff base
Online: 10 March 2017 (10:11:56 CET)
ARTICLE
|
doi:10.20944/preprints202403.0640.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
artemisinin; artesunate; dihydroartemisinin; artemether; Artemisia annua, Artemisia afra, tea infusion; α-SMA
Online: 11 March 2024 (18:08:23 CET)
ARTICLE
|
doi:10.20944/preprints202402.1663.v1
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
Silibinin; Silybin; Natural products; Mitsunobu reaction; Antioxidants; Human prostate cancer
Online: 29 February 2024 (08:22:17 CET)
ARTICLE
|
doi:10.20944/preprints201609.0123.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
carbonic anhydrase; acetylcholinesterase; β-Lactam; 2-Azetidinone; enzyme inhibition; enzyme purification
Online: 30 September 2016 (05:38:45 CEST)
REVIEW
|
doi:10.20944/preprints202402.0911.v1
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
indole alkaloids; marine resources; biological activity; therapeutic application; synthetic strategies
Online: 16 February 2024 (14:17:18 CET)
ARTICLE
|
doi:10.20944/preprints202104.0362.v1
Subject:
Computer Science And Mathematics,
Mathematics
Keywords:
Tempered Fractional Derivative; One-sided Tempered Fractional Derivative; Bilateral Tempered Fractional Derivative; Tempered Riesz potential.
Online: 13 April 2021 (18:48:08 CEST)
ARTICLE
|
doi:10.20944/preprints202405.1732.v1
Subject:
Medicinal Chemistry,
Chemistry And Materials Science
Keywords:
carbamates; oxamates; synthetic cytokinins; substituted ureas; anti-oxidative effect; cytotoxicity; oxidative stress
Online: 27 May 2024 (10:27:42 CEST)
ARTICLE
|
doi:10.20944/preprints202312.1717.v1
Subject:
Medicine And Pharmacology,
Other
Keywords:
Cordycepin derivatives; Antitumor; structural modification
Online: 22 December 2023 (08:09:53 CET)
ARTICLE
|
doi:10.20944/preprints202406.0319.v1
Subject:
Analysis,
Computer Science And Mathematics
Keywords:
Shift-invariant; Scale-invariant; Nabla derivative; Fractional q-derivative; Fractional Hahn derivative.
Online: 5 June 2024 (15:24:22 CEST)
ARTICLE
|
doi:10.20944/preprints201805.0040.v2
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
inhibiting activity; catalysis; cyclization; olivacine; palladium; pyrido[4,3-b]carbazoles
Online: 1 June 2018 (09:39:56 CEST)
REVIEW
|
doi:10.20944/preprints202310.1501.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
plant triterpenoid; structure modifier; antiviral activity; HIV-1; HSV-1; maturation inhibitor
Online: 24 October 2023 (07:33:45 CEST)
REVIEW
|
doi:10.20944/preprints202308.2076.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
monoterpene; pharmacophore; chemical modification; antiviral; anticancer; anxiolytic; neuroprotective activity
Online: 30 August 2023 (11:04:58 CEST)
REVIEW
|
doi:10.20944/preprints202212.0164.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
Fractional Derivative; Fractional Calculus; Machine Learning; Artificial Intelligence; Complexity; Regression Analysis
Online: 8 December 2022 (14:45:05 CET)
ARTICLE
|
doi:10.20944/preprints202008.0524.v1
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
Isoxazolines; nitrile oxide; 1,3-dipolar cycloaddition; antibacterial activity; antioxidant activity
Online: 24 August 2020 (10:03:22 CEST)
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
oleanolic acid derivatives; synthesis; anti-tumor activity; molecular docking; computer-aided drug design
Online: 24 April 2017 (12:08:36 CEST)
ARTICLE
|
doi:10.20944/preprints202401.0386.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
schiff bases; benitrobenrazide; benserazide; hexokinase 2; enzyme inhibition
Online: 4 January 2024 (12:30:49 CET)
ARTICLE
|
doi:10.20944/preprints201912.0099.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Leishmania; thiochromenes; benzothiopyrans; cytotoxicity
Online: 8 December 2019 (15:54:40 CET)
ARTICLE
|
doi:10.20944/preprints202311.0335.v1
Subject:
Chemistry And Materials Science,
Biomaterials
Keywords:
poly-3-hydroxybutyrate; chlorophyll derivatives; electrospinning; antibacterial properties; supramolecular structure
Online: 7 November 2023 (02:49:38 CET)
ARTICLE
|
doi:10.20944/preprints202310.0436.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
pharmacological evaluation; docking; anti-inflammatory; analgesic; antimicrobial
Online: 8 October 2023 (08:26:48 CEST)
ARTICLE
|
doi:10.20944/preprints202210.0398.v1
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
Perfluorinated derivatives; Nucleophilic Aromatic Substitution; Bioconjugation; IR and 19F-NMR simulations; Molecular Docking
Online: 26 October 2022 (04:01:55 CEST)
ARTICLE
|
doi:10.20944/preprints202103.0399.v1
Subject:
Engineering,
Automotive Engineering
Keywords:
Fractional derivative; Derivative order; Hermitian system; Complex order; Liouville derivative
Online: 15 March 2021 (16:23:56 CET)
ARTICLE
|
doi:10.20944/preprints202309.0262.v1
Subject:
Computer Science And Mathematics,
Mathematics
Keywords:
fractional calculus; difference-differential operator; special function
Online: 5 September 2023 (11:46:40 CEST)
ARTICLE
|
doi:10.20944/preprints202308.0877.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Quinolizidine derivatives; Lupinine, Cytisine; Sparteine; Antiarrhythmic activity; Inotropic and chronotropic activities; Vasorelaxant activity
Online: 11 August 2023 (03:03:24 CEST)
ARTICLE
|
doi:10.20944/preprints202210.0055.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
metapneumovirus; molecular docking; phenolic compounds; glycosides; ellagic acid; RNA-dependent RNA-polymerase
Online: 6 October 2022 (08:40:19 CEST)
ARTICLE
|
doi:10.20944/preprints201801.0023.v1
Subject:
Business, Economics And Management,
Finance
Keywords:
perturbation expansion; Green’s function; model risk; model uncertainty; credit derivatives; CVA; correlation risk
Online: 4 January 2018 (03:24:24 CET)
ARTICLE
|
doi:10.20944/preprints202401.0965.v2
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
1,2-(α -ketotetramethylene)-ferrocene; 1,2-(tetramethylene)-ferrocene; ferrocene; Friedel-Crafts acylation; Clemmensen reduction; X-ray crystallography; planar chirality; puckering parameters; electrochemistry
Online: 29 January 2024 (04:43:43 CET)
ARTICLE
|
doi:10.20944/preprints202311.0711.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
antifungal potential; naphthoquinone derivatives; 2,3-DBNQ; fungal membrane permeability; cytotoxicity
Online: 13 November 2023 (08:25:22 CET)
ARTICLE
|
doi:10.20944/preprints202304.0915.v1
Subject:
Engineering,
Civil Engineering
Keywords:
composite improved soil; expansive soil; lignin and its derivatives; mechanical properties; micro characteristics; improvement mechanis
Online: 25 April 2023 (09:57:31 CEST)
ARTICLE
|
doi:10.20944/preprints202304.0913.v1
Subject:
Engineering,
Civil Engineering
Keywords:
Composite improved soil; expansive soil; lignin and its derivatives; mechanical properties; micro characteristics; improvement mechanis
Online: 25 April 2023 (09:49:07 CEST)
ARTICLE
|
doi:10.20944/preprints201808.0463.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Factor Xa ( F-Xa), Cardiovascular diseases (CD), Coronary heart disease (CHD), Tissue plasminogen activator (t-PA), Urokinase (UK), Streptokinase (SK), N,N-Dimethyl formamide (DMF)
Online: 27 August 2018 (14:54:10 CEST)
ARTICLE
|
doi:10.20944/preprints202405.2011.v1
Subject:
Organic Chemistry,
Chemistry And Materials Science
Keywords:
pyridazine N-oxide; photoisomerization; DFT calculations; pyrazole; furan.
Online: 30 May 2024 (08:12:30 CEST)
REVIEW
|
doi:10.20944/preprints202401.0005.v1
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
Suzuki coupling; Stille coupling; Negishi coupling; Ullmann coupling; Wurtz coupling; electrochemical method
Online: 3 January 2024 (02:09:30 CET)
REVIEW
|
doi:10.20944/preprints202310.0625.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
anthracene derivatives; breast cancer; natural products; biological activity; emodin; aloe-emodin; hypericin; chrysophanol; rhein; physcion
Online: 11 October 2023 (04:46:44 CEST)
ARTICLE
|
doi:10.20944/preprints201901.0307.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
molecular docking; fluoroquinolones; antimicrobial activity
Online: 30 January 2019 (09:31:52 CET)
ARTICLE
|
doi:10.20944/preprints201804.0025.v1
Online: 2 April 2018 (11:27:27 CEST)
REVIEW
|
doi:10.20944/preprints202306.2174.v1
Subject:
Biology And Life Sciences,
Neuroscience And Neurology
Keywords:
Andrographis paniculata; Andrographolide; Neurodegenerative Diseases; Alzheimer; Parkinson; Brain Ischemia; Neuroinflammation
Online: 30 June 2023 (07:38:39 CEST)
REVIEW
|
doi:10.20944/preprints202403.0494.v1
Subject:
Dermatology,
Medicine And Pharmacology
Keywords:
xanthone, telangiectasia, rosacea, vascular disorders, cosmetics, dermatology, blood vessels
Online: 8 March 2024 (06:25:27 CET)
ARTICLE
|
doi:10.20944/preprints202312.1808.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
piperazine/morpholine derivatives; HRMS; MSn; structural characterization; antimicrobial activity.
Online: 25 December 2023 (08:20:57 CET)
ARTICLE
|
doi:10.20944/preprints202311.1837.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
1,3,5-triazine; nucleophilic substitution; nitrosation reaction; azido-acetylene cycloaddition; 1,2,3-triazole; hyperbranched polymers; antibacterial activity; cytotoxicity; M-HeLa; Vero
Online: 29 November 2023 (08:10:21 CET)
REVIEW
|
doi:10.20944/preprints202311.0160.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
pyrethrins; pyrethroids; insecticides; terpenoids; pyrethrum.
Online: 2 November 2023 (10:36:10 CET)
ARTICLE
|
doi:10.20944/preprints202305.1839.v2
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Anti-tubercular agents; DprE1 inhibitor; Structure activity relationship; in vivo activity
Online: 1 June 2023 (07:42:34 CEST)
ARTICLE
|
doi:10.20944/preprints201711.0177.v2
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Leishmania; thiochroman-4-ones; acyl hydrazone; cytotoxicity
Online: 2 January 2018 (10:11:55 CET)
ARTICLE
|
doi:10.20944/preprints202404.0478.v1
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
Xylaria sp.; pyranone derivative; sesquiterpenoid; antimicrobial activity
Online: 8 April 2024 (16:42:40 CEST)
ARTICLE
|
doi:10.20944/preprints202305.0228.v1
Subject:
Chemistry And Materials Science,
Physical Chemistry
Keywords:
rational design; antioxidants; electron transfer; hydrogen transfer; neuroprotection; AChE; COMT; MAOB
Online: 4 May 2023 (08:13:16 CEST)
ARTICLE
|
doi:10.20944/preprints202303.0502.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Tuberculosis; Biscoumarins; Ligand molecules; DprE1; Anti-tuberculosis activity; Molecular docking; MD Simulation; Cytotoxicity
Online: 29 March 2023 (04:21:45 CEST)
ARTICLE
|
doi:10.20944/preprints202210.0216.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
anti-inflammatory substance; N-acylhydrazone; naphthyl-N-acylhydrazone; LASSBio-1524 analogues
Online: 14 October 2022 (14:21:35 CEST)
ARTICLE
|
doi:10.20944/preprints202008.0438.v1
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
acetylcholinesterase; antioxidant; Alzheimer; coumarin; selenazole
Online: 20 August 2020 (07:26:34 CEST)
ARTICLE
|
doi:10.20944/preprints202002.0453.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Michael acceptor; safe covalent drugs; oxidative stress inducers; trans-cinnamaldehyde; curcumin; colorectal cancer
Online: 29 February 2020 (04:22:03 CET)
ARTICLE
|
doi:10.20944/preprints201902.0248.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
10-methoxycanthin-6-one; quaternization; antibacterial; SARs
Online: 27 February 2019 (05:08:02 CET)
ARTICLE
|
doi:10.20944/preprints201811.0330.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
hyperpigmentation; tyrosinase inhibitors; 3-(2,4-dihydroxyphenyl)propionic acid; structure-activity relationship study; B16-F10 cellular melanogenesis inhibition
Online: 14 November 2018 (09:59:45 CET)
ARTICLE
|
doi:10.20944/preprints201805.0196.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
P-glycoprotein; glioblastoma multiforme; brain-blood barrier; doxorubicin
Online: 14 May 2018 (12:50:18 CEST)
ARTICLE
|
doi:10.20944/preprints202312.0898.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
triazinyl phosphoramidate; amphiphilic oligonucleotides; self-assembly; human serum albumin; Ku antigen; PARP1; protein-oligonucleotide complexes
Online: 12 December 2023 (13:53:44 CET)
ARTICLE
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
(S)-Practolol; paracetamol; (S)-pindolol; (S)-carteolol; Candida antarctica Lipase B; chiral chromatography; dimer formation
Online: 4 March 2021 (08:34:02 CET)
ARTICLE
|
doi:10.20944/preprints202007.0056.v1
Subject:
Chemistry And Materials Science,
Materials Science And Technology
Keywords:
Aggregation-induced emission; quinones; fluorescence; TD-DFT; quantum yield
Online: 5 July 2020 (08:38:20 CEST)
BRIEF REPORT
|
doi:10.20944/preprints202001.0292.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
circadian rhythms; small molecules; luciferase reporters; period estimations
Online: 25 January 2020 (00:33:40 CET)
ARTICLE
|
doi:10.20944/preprints202311.0516.v1
Subject:
Computer Science And Mathematics,
Other
Keywords:
fuzzy set; intuitionistic fuzzy number; Hukuhara differentiable; generalized Hukuhara differentiable
Online: 8 November 2023 (04:49:07 CET)
ARTICLE
|
doi:10.20944/preprints202305.1517.v2
Subject:
Biology And Life Sciences,
Virology
Keywords:
Antiviral; Thiourea derivatives; Hepatitis B Virus; Chronic hepatitis B infection; Mitochondria dysfunction; Exhausted hepatocytes
Online: 29 May 2023 (14:29:16 CEST)
ARTICLE
|
doi:10.20944/preprints202304.0730.v1
Subject:
Physical Sciences,
Optics And Photonics
Keywords:
Near infrared emission; Aza-Bodipy derivatives; Saturable absorption; Nonlinear refraction; Two-photon absorption
Online: 23 April 2023 (02:41:33 CEST)
ARTICLE
|
doi:10.20944/preprints202301.0290.v1
Subject:
Computer Science And Mathematics,
Analysis
Keywords:
generalized Sonin condition; general fractional integral; general fractional derivative of arbitrary order; regularized general fractional derivative of arbitrary order; 1st level general fractional derivative; 1st fundamental theorem of fractional calculus; 2nd fundamental theorem of fractional calculus
Online: 17 January 2023 (01:34:12 CET)
REVIEW
|
doi:10.20944/preprints202211.0271.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
cisplatin; carboplatin; oxaliplatin; cellular uptake; DNA damage; transcription regulation; non-nuclear targets; chemoresistance; mechanisms of action; clinical usages; influx and efflux pumps; ribosome biogenesis; ER stress response; immunogenic cell death; interstrand and intrastrand DNA cross-links.
Online: 15 November 2022 (03:38:06 CET)
ARTICLE
|
doi:10.20944/preprints202401.1785.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Synthesis; In silico; In vitro; Phenothiazine; Sulphonamide; Antimicrobial
Online: 24 January 2024 (15:38:29 CET)
ARTICLE
|
doi:10.20944/preprints202308.1350.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Imidazole; Imidazole derivative; Sirtuins; NSCLC; Epigenetics
Online: 18 August 2023 (09:04:18 CEST)
ARTICLE
|
doi:10.20944/preprints202304.1201.v1
Subject:
Biology And Life Sciences,
Insect Science
Keywords:
Insecta; pest control; ecotoxicology; behavior; biological products; germoplasm; essential oil; insecticide; necrophoresis
Online: 29 April 2023 (04:06:06 CEST)
ARTICLE
|
doi:10.20944/preprints202102.0608.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
Cape Verde; cereals; metals; dietary intake; risk evaluation
Online: 26 February 2021 (11:05:17 CET)
ARTICLE
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
myricetin; ferulic acid; antiviral activity; microscale thermophoresis; molecular docking
Online: 24 November 2019 (16:29:54 CET)
ARTICLE
|
doi:10.20944/preprints201901.0086.v1
Subject:
Business, Economics And Management,
Finance
Keywords:
Quinoxaline Analogs, Synthesis, Thymidine phosphorylase inhibition, Molecular docking
Online: 9 January 2019 (13:23:49 CET)
ARTICLE
|
doi:10.20944/preprints202401.1031.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
antiproliferative activity; amines; amides; benzimidazoles; interaction with DNA
Online: 12 January 2024 (15:11:23 CET)
REVIEW
|
doi:10.20944/preprints202312.1484.v1
Subject:
Chemistry And Materials Science,
Inorganic And Nuclear Chemistry
Keywords:
antibacterial activities; cytotoxic properties; uracil; 6-methyl-2-thiouracil; 6-propyl-2-thiouracil; 2-thiouracil
Online: 20 December 2023 (07:12:54 CET)
ARTICLE
|
doi:10.20944/preprints202307.0765.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
4-amino-7-chloroquinoline; 1,3,4-oxadiazole; anthranilic acid; synthesis; quorum sensing; anti-biofilm; P. aeruginosa; PQS
Online: 12 July 2023 (21:25:14 CEST)
ARTICLE
|
doi:10.20944/preprints202304.0220.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
breast cancer; cervical cancer; stem cells; docking; simulation; microRNA
Online: 11 April 2023 (10:14:48 CEST)
ARTICLE
|
doi:10.20944/preprints202403.0635.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
azaphenothiazine; chlorpromazine; quinobenzothiazine; anticancer activity; antibacterial activity; apoptotic activity; cell cycle arrest
Online: 12 March 2024 (04:26:43 CET)
ARTICLE
|
doi:10.20944/preprints202109.0311.v1
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
Quinazolinone; Styrene; Methacrylate; Nano-silver; Antibacterial; Antitumor.
Online: 17 September 2021 (12:11:48 CEST)
ARTICLE
|
doi:10.20944/preprints201904.0262.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
total synthesis; antitumor activity; structure-activity relationship
Online: 24 April 2019 (05:29:48 CEST)
ARTICLE
|
doi:10.20944/preprints201801.0260.v1
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
Acylhydrazone; Pyrazole; X-ray crystallography; DFT/B3LYP; Catecholase activity
Online: 28 January 2018 (12:44:49 CET)
ARTICLE
|
doi:10.20944/preprints201710.0200.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
4-Thiazolidinones; ORAC assay; Metalloproteinase-9; Docking study; Keratinocytes cultures; Nuclear factor -kB.
Online: 31 October 2017 (16:36:16 CET)
REVIEW
|
doi:10.20944/preprints202401.1759.v1
Subject:
Chemistry And Materials Science,
Electronic, Optical And Magnetic Materials
Keywords:
Donor-acceptor-donor (D-A-D) derivatives; organic light emitting diode (OLED); high efficiency; emission; thermal analysis; synthesis.
Online: 24 January 2024 (10:38:10 CET)
BRIEF REPORT
|
doi:10.20944/preprints202401.0128.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Psoralen; Calf-thymus; Oligo (dAdT); Fluorometry; 8-Methoxypsoralen (8-MOP); Aminomethlytrimethylpsoralen (AMT); 6E; Photochemotherapy; Binding; Scatchard; DNA (AT-40)
Online: 3 January 2024 (05:40:18 CET)
ARTICLE
|
doi:10.20944/preprints201805.0073.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
cancer treatment; chlorin; Photodynamic therapy (PDT); photosensitizer; tumor size
Online: 3 May 2018 (12:16:15 CEST)
ARTICLE
|
doi:10.20944/preprints202306.0167.v1
Subject:
Chemistry And Materials Science,
Applied Chemistry
Keywords:
1,2-Diphenyl-o-carborane; Chromium Metal Complexes; Boron Neutron Capture Therapy; Biological Evaluation; Cytotoxicity
Online: 2 June 2023 (09:18:49 CEST)
REVIEW
|
doi:10.20944/preprints202305.2171.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
caffeic acid phenethyl ester; CAPE derivatives; anti-inflammatory; NF-kB; antioxidant; Nrf2; neuroprotection
Online: 31 May 2023 (05:32:19 CEST)
ARTICLE
|
doi:10.20944/preprints201611.0072.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
aporphine derivatives; antiarrhythmia; 10,11-dibromocrebanine; 3-bromocrebanine; crebanine; stephanine
Online: 14 November 2016 (07:24:04 CET)
ARTICLE
|
doi:10.20944/preprints202210.0368.v1
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
anabasine; amides; quaternary pyridinium salts; isoxazole; isothiazole; pyridine; adamantane; antiviral activity; antimicrobial activity; analgesic activity; cytisine
Online: 24 October 2022 (13:58:21 CEST)
ARTICLE
|
doi:10.20944/preprints202309.1706.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
isoxazolidine derivatives; 1,3-dipolar cycloaddition; α-aryl-N-methyl nitrones; Density Functional Theory (DFT); Electron Localization Function (ELF); CDFT indices; docking; molecular dynamics; EGFR; binding energy
Online: 26 September 2023 (04:37:56 CEST)
REVIEW
|
doi:10.20944/preprints202308.1553.v1
Online: 22 August 2023 (10:10:52 CEST)
ARTICLE
|
doi:10.20944/preprints202305.0222.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Amino acid derivatives; Digestive enzymes; Pancreatic lipase; Pancreatic α-Amylase; α-Glucosidase; Metabolic disorders
Online: 4 May 2023 (07:59:29 CEST)
ARTICLE
|
doi:10.20944/preprints202201.0359.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
JAK/STAT3 signaling pathway; Meridianin derivatives; Isothiouronium; Anti-tumor activity
Online: 24 January 2022 (14:06:38 CET)
ARTICLE
|
doi:10.20944/preprints202011.0416.v2
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
LD50; lethal Dose; Xylometazoline; Oxymetazoline; Imidazoline Derivatives
Online: 15 December 2020 (13:03:01 CET)
ARTICLE
|
doi:10.20944/preprints202001.0081.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Berberine; Lipophilic substituent; Anti-cancer activity; Photocytotoxicity; Reactive oxygen species
Online: 9 January 2020 (11:30:40 CET)
ARTICLE
|
doi:10.20944/preprints201704.0032.v1
Subject:
Chemistry And Materials Science,
Chemical Engineering
Keywords:
Olefin metathesis; ethyl linoleate; ruthenium
Online: 5 April 2017 (18:22:30 CEST)
ARTICLE
|
doi:10.20944/preprints202312.2085.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Dermaseptin B2; Dermaseptin S4; analogs; Acinetobacter baumannii; Healthcare-Associated Infections; Antibacterial activity
Online: 27 December 2023 (10:24:49 CET)
ARTICLE
|
doi:10.20944/preprints202304.0369.v1
Subject:
Business, Economics And Management,
Econometrics And Statistics
Keywords:
Deep learning; Backward stochastic differential equation; Nonlinear Feynman-Kac formula; High dimensional PDE; Derivatives pricing; Neural network
Online: 14 April 2023 (10:44:44 CEST)
ARTICLE
|
doi:10.20944/preprints202206.0188.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Stigmatellin; Myxobacteria; Biosynthesis; Natural Products; Secondary Metabolites
Online: 13 June 2022 (12:58:42 CEST)
ARTICLE
|
doi:10.20944/preprints202206.0099.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
Chitosan; mHTCC; SARS-CoV-2; S protein; ACE2; Molecular interaction
Online: 7 June 2022 (09:05:16 CEST)
ARTICLE
|
doi:10.20944/preprints202201.0475.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
DAST; semi-synthesis; fluorination; Beckmann-rearrangement; cyclopropane; natural product; ecdysteroid; NMR; structure elucidation; anticancer
Online: 31 January 2022 (21:35:38 CET)