Search Results
34599 articles found
ARTICLE
|
doi:10.20944/preprints202406.0319.v1
Subject:
Computer Science And Mathematics,
Analysis
Keywords:
Shift-invariant; Scale-invariant; Nabla derivative; Fractional q-derivative; Fractional Hahn derivative.
Online: 5 June 2024 (15:24:22 CEST)
ARTICLE
|
doi:10.20944/preprints202406.0843.v1
Subject:
Engineering,
Marine Engineering
Keywords:
Wave energy converter; Oscillation; Wave force; Wave-structure interaction; Water waves
Online: 12 June 2024 (15:04:16 CEST)
ARTICLE
|
doi:10.20944/preprints202404.0444.v1
Subject:
Engineering,
Transportation Science And Technology
Keywords:
submarine; stern rudder -plane configuration; rudder force and moment; RANS-based simulation
Online: 7 April 2024 (13:59:38 CEST)
ARTICLE
|
doi:10.20944/preprints202404.0439.v1
Subject:
Environmental And Earth Sciences,
Pollution
Keywords:
eutrophication; phytoplankton blooms; Sentinel-2; hydrodynamic modelling; Pilica River; Sulejow Reservoir; NDCl; CCHE2D
Online: 5 April 2024 (12:09:49 CEST)
ARTICLE
|
doi:10.20944/preprints201610.0079.v1
Subject:
Engineering,
Civil Engineering
Keywords:
river confluence; stage-discharge relationship; hydrodynamic influence; backwater; flow separation
Online: 19 October 2016 (12:31:32 CEST)
ARTICLE
|
doi:10.20944/preprints202406.1337.v1
Subject:
Environmental And Earth Sciences,
Water Science And Technology
Keywords:
electrochemical bioassay; mediator; Escherichia coli; hydrodynamic voltammetry; antibiotics
Online: 20 June 2024 (04:43:25 CEST)
ARTICLE
|
doi:10.20944/preprints201908.0299.v1
Subject:
Environmental And Earth Sciences,
Oceanography
Keywords:
Istanbul Strait; stratified flow; gravity driven flow; numerical modelling
Online: 28 August 2019 (15:23:55 CEST)
ARTICLE
|
doi:10.20944/preprints202403.1557.v1
Subject:
Chemistry And Materials Science,
Polymers And Plastics
Keywords:
biodegradable polymers; antibacterial polymers; chitosan Schiff base; κ-carrageenan blend; grafted copolymer
Online: 26 March 2024 (11:30:13 CET)
ARTICLE
|
doi:10.20944/preprints202403.0479.v1
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
quinone; quinone imine; hydrogen bonding; X-ray crystallography; NMR titration; redox.
Online: 8 March 2024 (10:33:48 CET)
ARTICLE
|
doi:10.20944/preprints202405.2011.v1
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
pyridazine N-oxide; photoisomerization; DFT calculations; pyrazole; furan.
Online: 30 May 2024 (08:12:30 CEST)
ARTICLE
|
doi:10.20944/preprints201805.0420.v1
Subject:
Physical Sciences,
Fluids And Plasmas Physics
Keywords:
wet agglomeration; flocculation; hydrodynamics; turbulence
Online: 29 May 2018 (09:00:36 CEST)
ARTICLE
|
doi:10.20944/preprints202403.0382.v1
Subject:
Chemistry And Materials Science,
Materials Science And Technology
Keywords:
donor-acceptor derivatives; blue organic light emitting diode; high efficiency; blue emission; thermal analysis
Online: 7 March 2024 (09:34:59 CET)
ARTICLE
|
doi:10.20944/preprints202403.0156.v1
Subject:
Engineering,
Energy And Fuel Technology
Keywords:
cattle manure; milking station; anaerobic digestion; pretreatment; hydrodynamic cavitation; biogas; methane; energy efficiency
Online: 6 March 2024 (04:05:53 CET)
COMMUNICATION
|
doi:10.20944/preprints202406.1464.v1
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
photosensitizers; photoredox catalysis; porphyrins; redox potential; substituent effects.
Online: 21 June 2024 (13:35:38 CEST)
ARTICLE
|
doi:10.20944/preprints201605.0002.v1
Online: 11 May 2016 (07:42:45 CEST)
ARTICLE
|
doi:10.20944/preprints202406.0049.v1
Subject:
Engineering,
Bioengineering
Keywords:
hydrodynamic resistance; microfluidics; differential pressure; metrology; test method
Online: 3 June 2024 (07:49:10 CEST)
ARTICLE
|
doi:10.20944/preprints201906.0043.v1
Subject:
Engineering,
Industrial And Manufacturing Engineering
Keywords:
microalgae; photobioreactor; flashing light effect; Computational Fluid Dynamics
Online: 5 June 2019 (14:56:44 CEST)
ARTICLE
|
doi:10.20944/preprints201611.0102.v1
Subject:
Engineering,
Marine Engineering
Keywords:
ocean wave energy; fluid-structure interaction; BEM; diffraction/ radiation; floating cylinder; heave; array
Online: 19 November 2016 (05:20:36 CET)
ARTICLE
|
doi:10.20944/preprints202008.0675.v1
Subject:
Environmental And Earth Sciences,
Geophysics And Geology
Keywords:
wave impact assessment; characteristic wave height; Salento peninsula; Taranto Gulf; Mediterranean Sea; November 2019 storm
Online: 30 August 2020 (15:53:07 CEST)
ARTICLE
|
doi:10.20944/preprints202309.2116.v1
Subject:
Engineering,
Marine Engineering
Keywords:
Wave power generation; Oscillating float; Computational Fluid Dynamics; Array
Online: 30 September 2023 (07:55:14 CEST)
ARTICLE
|
doi:10.20944/preprints202003.0263.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
pectin; antibacterial; lemon; flavonoids; hydrodynamic cavitation; IntegroPectin
Online: 17 March 2020 (03:43:39 CET)
ARTICLE
|
doi:10.20944/preprints201703.0053.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
1,3,4-Thiadiazole; 1,2,4-Triazole; synthesis; MTT assay; Cytotoxicity of Schiff base
Online: 10 March 2017 (10:11:56 CET)
ARTICLE
|
doi:10.20944/preprints202402.0887.v1
Subject:
Chemistry And Materials Science,
Materials Science And Technology
Keywords:
Calixarene; Dihomooxacalixarene; Hexahomotrioxacalixarene; Pseudopolymorphism; X-ray diffraction
Online: 16 February 2024 (06:58:09 CET)
ARTICLE
|
doi:10.20944/preprints202405.0491.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Acetaminophen; Benzothiazoles; Azo dyes; Shigella flexneri; Anti-Shigella activity; Repositioning; Combination studies; Diarrhea.
Online: 8 May 2024 (11:33:24 CEST)
ARTICLE
|
doi:10.20944/preprints202301.0167.v1
Subject:
Chemistry And Materials Science,
Food Chemistry
Keywords:
Almond; Almond beverage; Almond skin; Antiradical activity; Green extraction; Hydrodynamic cavitation; Nutritional values; Polyphenols; Proteins; Vitamins
Online: 10 January 2023 (02:12:56 CET)
ARTICLE
|
doi:10.20944/preprints201907.0325.v1
Subject:
Chemistry And Materials Science,
Food Chemistry
Keywords:
biomethane; d-limonene; flavanones; food waste; green extraction; hydrodynamic cavitation; orange waste; pectin; polyphenols
Online: 29 July 2019 (04:04:30 CEST)
REVIEW
|
doi:10.20944/preprints202407.0170.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Glycerol; Solketal; alkylglycerol; organochalcogen; green-solvent; glycidol
Online: 2 July 2024 (09:46:04 CEST)
ARTICLE
|
doi:10.20944/preprints202104.0362.v1
Subject:
Computer Science And Mathematics,
Mathematics
Keywords:
Tempered Fractional Derivative; One-sided Tempered Fractional Derivative; Bilateral Tempered Fractional Derivative; Tempered Riesz potential.
Online: 13 April 2021 (18:48:08 CEST)
ARTICLE
|
doi:10.20944/preprints202404.1360.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
ovarian cancer; 2C; apoptosis; E2F1, in silico docking.
Online: 19 April 2024 (16:08:57 CEST)
REVIEW
|
doi:10.20944/preprints202403.0494.v1
Subject:
Medicine And Pharmacology,
Dermatology
Keywords:
xanthone, telangiectasia, rosacea, vascular disorders, cosmetics, dermatology, blood vessels
Online: 8 March 2024 (06:25:27 CET)
ARTICLE
|
doi:10.20944/preprints202001.0266.v1
Subject:
Engineering,
Civil Engineering
Keywords:
rubble-mound; zero-freeboard; porous-media; immersed-boundary; level-set; Smagorinsky subgrid scale model; wave reflection; wave transmission; wave overtopping; wave setup
Online: 23 January 2020 (14:43:47 CET)
ARTICLE
|
doi:10.20944/preprints201809.0574.v1
Subject:
Engineering,
Chemical Engineering
Keywords:
hydrodynamic; gas retention; submerged membrane bioreactor; influence of temperature; oxygen mass transfer coefficient
Online: 29 September 2018 (03:53:05 CEST)
ARTICLE
|
doi:10.20944/preprints201803.0088.v1
Subject:
Engineering,
Civil Engineering
Keywords:
extreme water level; hydrodynamic model; Monte Carlo; joint probability; model calibration and verification; Danshuei River system
Online: 12 March 2018 (07:56:58 CET)
ARTICLE
|
doi:10.20944/preprints202001.0157.v3
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
pectin; antioxidant; lemon; flavonoids; hydrodynamic cavitation; IntegroPectin
Online: 31 March 2020 (05:00:13 CEST)
ARTICLE
|
doi:10.20944/preprints202407.0929.v1
Subject:
Chemistry And Materials Science,
Inorganic And Nuclear Chemistry
Keywords:
antimicrobial activity; copper(II) complexes; 2,4-dithiouracil; gold(III) complexes
Online: 12 July 2024 (09:39:49 CEST)
ARTICLE
|
doi:10.20944/preprints202403.0640.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
artemisinin; artesunate; dihydroartemisinin; artemether; Artemisia annua, Artemisia afra, tea infusion; α-SMA
Online: 11 March 2024 (18:08:23 CET)
REVIEW
|
doi:10.20944/preprints202402.0911.v1
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
indole alkaloids; marine resources; biological activity; therapeutic application; synthetic strategies
Online: 16 February 2024 (14:17:18 CET)
ARTICLE
|
doi:10.20944/preprints202312.1717.v1
Subject:
Medicine And Pharmacology,
Other
Keywords:
Cordycepin derivatives; Antitumor; structural modification
Online: 22 December 2023 (08:09:53 CET)
ARTICLE
|
doi:10.20944/preprints202402.1663.v1
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
Silibinin; Silybin; Natural products; Mitsunobu reaction; Antioxidants; Human prostate cancer
Online: 29 February 2024 (08:22:17 CET)
ARTICLE
|
doi:10.20944/preprints201609.0123.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
carbonic anhydrase; acetylcholinesterase; β-Lactam; 2-Azetidinone; enzyme inhibition; enzyme purification
Online: 30 September 2016 (05:38:45 CEST)
ARTICLE
|
doi:10.20944/preprints202406.0465.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
betulonic acid; triterpenoid; lupan; natural product; chemical transformation; synthesis; spectroscopic method; cytotoxicity; antimicrobial activity
Online: 7 June 2024 (07:57:23 CEST)
ARTICLE
|
doi:10.20944/preprints201805.0040.v2
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
inhibiting activity; catalysis; cyclization; olivacine; palladium; pyrido[4,3-b]carbazoles
Online: 1 June 2018 (09:39:56 CEST)
REVIEW
|
doi:10.20944/preprints202310.1501.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
plant triterpenoid; structure modifier; antiviral activity; HIV-1; HSV-1; maturation inhibitor
Online: 24 October 2023 (07:33:45 CEST)
REVIEW
|
doi:10.20944/preprints202308.2076.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
monoterpene; pharmacophore; chemical modification; antiviral; anticancer; anxiolytic; neuroprotective activity
Online: 30 August 2023 (11:04:58 CEST)
REVIEW
|
doi:10.20944/preprints202212.0164.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
Fractional Derivative; Fractional Calculus; Machine Learning; Artificial Intelligence; Complexity; Regression Analysis
Online: 8 December 2022 (14:45:05 CET)
ARTICLE
|
doi:10.20944/preprints202008.0524.v1
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
Isoxazolines; nitrile oxide; 1,3-dipolar cycloaddition; antibacterial activity; antioxidant activity
Online: 24 August 2020 (10:03:22 CEST)
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
oleanolic acid derivatives; synthesis; anti-tumor activity; molecular docking; computer-aided drug design
Online: 24 April 2017 (12:08:36 CEST)
ARTICLE
|
doi:10.20944/preprints202406.0032.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
HIV-1; reverse transcriptase; polymerase; ribonuclease H; inhibitor; benzisothiazolone
Online: 3 June 2024 (07:56:06 CEST)
ARTICLE
Subject:
Chemistry And Materials Science,
Biomaterials
Keywords:
Polymer Nanocomposites; Nanofiller Dispersion; Flow-Cells; Experimental and Numerical; Viscoelastic Fluids
Online: 1 December 2020 (18:25:01 CET)
ARTICLE
|
doi:10.20944/preprints202405.1732.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
carbamates; oxamates; synthetic cytokinins; substituted ureas; anti-oxidative effect; cytotoxicity; oxidative stress
Online: 27 May 2024 (10:27:42 CEST)
ARTICLE
|
doi:10.20944/preprints202401.0386.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
schiff bases; benitrobenrazide; benserazide; hexokinase 2; enzyme inhibition
Online: 4 January 2024 (12:30:49 CET)
ARTICLE
|
doi:10.20944/preprints201912.0099.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Leishmania; thiochromenes; benzothiopyrans; cytotoxicity
Online: 8 December 2019 (15:54:40 CET)
ARTICLE
|
doi:10.20944/preprints202311.0335.v1
Subject:
Chemistry And Materials Science,
Biomaterials
Keywords:
poly-3-hydroxybutyrate; chlorophyll derivatives; electrospinning; antibacterial properties; supramolecular structure
Online: 7 November 2023 (02:49:38 CET)
ARTICLE
|
doi:10.20944/preprints202310.0436.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
pharmacological evaluation; docking; anti-inflammatory; analgesic; antimicrobial
Online: 8 October 2023 (08:26:48 CEST)
ARTICLE
|
doi:10.20944/preprints202210.0398.v1
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
Perfluorinated derivatives; Nucleophilic Aromatic Substitution; Bioconjugation; IR and 19F-NMR simulations; Molecular Docking
Online: 26 October 2022 (04:01:55 CEST)
ARTICLE
|
doi:10.20944/preprints202103.0399.v1
Subject:
Engineering,
Automotive Engineering
Keywords:
Fractional derivative; Derivative order; Hermitian system; Complex order; Liouville derivative
Online: 15 March 2021 (16:23:56 CET)
ARTICLE
|
doi:10.20944/preprints202303.0417.v1
Subject:
Environmental And Earth Sciences,
Soil Science
Keywords:
Coastal flow slides; critical angle; retrogressive breach failure; hydrodynamic sediment transport; Monte Carlo simulation; risk assessment
Online: 23 March 2023 (14:47:06 CET)
ARTICLE
|
doi:10.20944/preprints202406.0056.v2
Subject:
Chemistry And Materials Science,
Materials Science And Technology
Keywords:
thiosemicarbazones; biodiesel; oxidative stability; kinetic study; energy
Online: 27 June 2024 (08:05:52 CEST)
ARTICLE
|
doi:10.20944/preprints202311.0889.v1
Subject:
Environmental And Earth Sciences,
Geography
Keywords:
anastomosing river; hydrodynamic parameters; calculation method; shape factor; scale factor; gradient factor
Online: 14 November 2023 (10:35:46 CET)
ARTICLE
|
doi:10.20944/preprints202309.0262.v1
Subject:
Computer Science And Mathematics,
Mathematics
Keywords:
fractional calculus; difference-differential operator; special function
Online: 5 September 2023 (11:46:40 CEST)
ARTICLE
|
doi:10.20944/preprints202308.0877.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Quinolizidine derivatives; Lupinine, Cytisine; Sparteine; Antiarrhythmic activity; Inotropic and chronotropic activities; Vasorelaxant activity
Online: 11 August 2023 (03:03:24 CEST)
ARTICLE
|
doi:10.20944/preprints202210.0055.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
metapneumovirus; molecular docking; phenolic compounds; glycosides; ellagic acid; RNA-dependent RNA-polymerase
Online: 6 October 2022 (08:40:19 CEST)
ARTICLE
|
doi:10.20944/preprints201801.0023.v1
Subject:
Business, Economics And Management,
Finance
Keywords:
perturbation expansion; Green’s function; model risk; model uncertainty; credit derivatives; CVA; correlation risk
Online: 4 January 2018 (03:24:24 CET)
ARTICLE
|
doi:10.20944/preprints202401.0965.v2
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
1,2-(α -ketotetramethylene)-ferrocene; 1,2-(tetramethylene)-ferrocene; ferrocene; Friedel-Crafts acylation; Clemmensen reduction; X-ray crystallography; planar chirality; puckering parameters; electrochemistry
Online: 29 January 2024 (04:43:43 CET)
ARTICLE
|
doi:10.20944/preprints201712.0005.v1
Subject:
Environmental And Earth Sciences,
Remote Sensing
Keywords:
Cloudburst; GIS; MIKE11; DEM; Hydrodynamic model
Online: 1 December 2017 (10:33:45 CET)
ARTICLE
|
doi:10.20944/preprints202405.1576.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
acetylenic; alkylglycerol; lipid0; solketal; shark liver oil
Online: 23 May 2024 (16:47:59 CEST)
ARTICLE
|
doi:10.20944/preprints202311.0711.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
antifungal potential; naphthoquinone derivatives; 2,3-DBNQ; fungal membrane permeability; cytotoxicity
Online: 13 November 2023 (08:25:22 CET)
ARTICLE
|
doi:10.20944/preprints202304.0915.v1
Subject:
Engineering,
Civil Engineering
Keywords:
composite improved soil; expansive soil; lignin and its derivatives; mechanical properties; micro characteristics; improvement mechanis
Online: 25 April 2023 (09:57:31 CEST)
ARTICLE
|
doi:10.20944/preprints202304.0913.v1
Subject:
Engineering,
Civil Engineering
Keywords:
Composite improved soil; expansive soil; lignin and its derivatives; mechanical properties; micro characteristics; improvement mechanis
Online: 25 April 2023 (09:49:07 CEST)
ARTICLE
|
doi:10.20944/preprints201808.0463.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Factor Xa ( F-Xa), Cardiovascular diseases (CD), Coronary heart disease (CHD), Tissue plasminogen activator (t-PA), Urokinase (UK), Streptokinase (SK), N,N-Dimethyl formamide (DMF)
Online: 27 August 2018 (14:54:10 CEST)
ARTICLE
|
doi:10.20944/preprints202406.0629.v1
Subject:
Physical Sciences,
Biophysics
Keywords:
individual molecule tracking; individual molecule; single molecule; diffusion; thermodynamic jitter; live cell; cytoplasm; liquids; room temperature; continuous-time random walk (CTRW); Brownian motion; anomalous motion; computer simulation
Online: 11 June 2024 (08:12:32 CEST)
ARTICLE
|
doi:10.20944/preprints202405.0395.v1
Subject:
Physical Sciences,
Biophysics
Keywords:
Individual molecule tracking; diffusion; thermodynamic jitter; live cell, cytoplasm, liquids, room temperature, continuous-time random walk (CTRW); Brownian motion/diffusion anomalous motion/diffusion; computer simulations
Online: 7 May 2024 (13:08:33 CEST)
REVIEW
|
doi:10.20944/preprints202401.0005.v1
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
Suzuki coupling; Stille coupling; Negishi coupling; Ullmann coupling; Wurtz coupling; electrochemical method
Online: 3 January 2024 (02:09:30 CET)
REVIEW
|
doi:10.20944/preprints202310.0625.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
anthracene derivatives; breast cancer; natural products; biological activity; emodin; aloe-emodin; hypericin; chrysophanol; rhein; physcion
Online: 11 October 2023 (04:46:44 CEST)
ARTICLE
|
doi:10.20944/preprints201901.0307.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
molecular docking; fluoroquinolones; antimicrobial activity
Online: 30 January 2019 (09:31:52 CET)
ARTICLE
|
doi:10.20944/preprints201804.0025.v1
Online: 2 April 2018 (11:27:27 CEST)
REVIEW
|
doi:10.20944/preprints202306.2174.v1
Subject:
Biology And Life Sciences,
Neuroscience And Neurology
Keywords:
Andrographis paniculata; Andrographolide; Neurodegenerative Diseases; Alzheimer; Parkinson; Brain Ischemia; Neuroinflammation
Online: 30 June 2023 (07:38:39 CEST)
ARTICLE
|
doi:10.20944/preprints201812.0175.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
Abies Alba Mill.; antioxidant activity; coniferous trees; essential oils; flavonoids; food preservation; green extraction; hydrodynamic cavitation; nutraceutics; polyphenols
Online: 17 December 2018 (07:07:56 CET)
BRIEF REPORT
|
doi:10.20944/preprints202111.0081.v1
Subject:
Environmental And Earth Sciences,
Atmospheric Science And Meteorology
Keywords:
electric streamer discharges; streamer theory; streamer parameters; plasma instabilities; partially-ionized plasmas; atmospheric electricity
Online: 3 November 2021 (13:59:43 CET)
ARTICLE
|
doi:10.20944/preprints202003.0128.v1
Subject:
Chemistry And Materials Science,
Metals, Alloys And Metallurgy
Keywords:
anisotropic yield criterion; hydrodynamic deep drawing; critical process window; aluminum alloy
Online: 8 March 2020 (04:03:25 CET)
ARTICLE
|
doi:10.20944/preprints202312.1808.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
piperazine/morpholine derivatives; HRMS; MSn; structural characterization; antimicrobial activity.
Online: 25 December 2023 (08:20:57 CET)
ARTICLE
|
doi:10.20944/preprints202311.1837.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
1,3,5-triazine; nucleophilic substitution; nitrosation reaction; azido-acetylene cycloaddition; 1,2,3-triazole; hyperbranched polymers; antibacterial activity; cytotoxicity; M-HeLa; Vero
Online: 29 November 2023 (08:10:21 CET)
REVIEW
|
doi:10.20944/preprints202311.0160.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
pyrethrins; pyrethroids; insecticides; terpenoids; pyrethrum.
Online: 2 November 2023 (10:36:10 CET)
ARTICLE
|
doi:10.20944/preprints202305.1839.v2
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Anti-tubercular agents; DprE1 inhibitor; Structure activity relationship; in vivo activity
Online: 1 June 2023 (07:42:34 CEST)
ARTICLE
|
doi:10.20944/preprints201711.0177.v2
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Leishmania; thiochroman-4-ones; acyl hydrazone; cytotoxicity
Online: 2 January 2018 (10:11:55 CET)
ARTICLE
|
doi:10.20944/preprints202404.0478.v1
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
Xylaria sp.; pyranone derivative; sesquiterpenoid; antimicrobial activity
Online: 8 April 2024 (16:42:40 CEST)
ARTICLE
|
doi:10.20944/preprints202305.0228.v1
Subject:
Chemistry And Materials Science,
Physical Chemistry
Keywords:
rational design; antioxidants; electron transfer; hydrogen transfer; neuroprotection; AChE; COMT; MAOB
Online: 4 May 2023 (08:13:16 CEST)
ARTICLE
|
doi:10.20944/preprints202303.0502.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Tuberculosis; Biscoumarins; Ligand molecules; DprE1; Anti-tuberculosis activity; Molecular docking; MD Simulation; Cytotoxicity
Online: 29 March 2023 (04:21:45 CEST)
ARTICLE
|
doi:10.20944/preprints202210.0216.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
anti-inflammatory substance; N-acylhydrazone; naphthyl-N-acylhydrazone; LASSBio-1524 analogues
Online: 14 October 2022 (14:21:35 CEST)
ARTICLE
|
doi:10.20944/preprints202008.0438.v1
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
acetylcholinesterase; antioxidant; Alzheimer; coumarin; selenazole
Online: 20 August 2020 (07:26:34 CEST)
ARTICLE
|
doi:10.20944/preprints202002.0453.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Michael acceptor; safe covalent drugs; oxidative stress inducers; trans-cinnamaldehyde; curcumin; colorectal cancer
Online: 29 February 2020 (04:22:03 CET)
ARTICLE
|
doi:10.20944/preprints201902.0248.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
10-methoxycanthin-6-one; quaternization; antibacterial; SARs
Online: 27 February 2019 (05:08:02 CET)
ARTICLE
|
doi:10.20944/preprints201811.0330.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
hyperpigmentation; tyrosinase inhibitors; 3-(2,4-dihydroxyphenyl)propionic acid; structure-activity relationship study; B16-F10 cellular melanogenesis inhibition
Online: 14 November 2018 (09:59:45 CET)
ARTICLE
|
doi:10.20944/preprints201805.0196.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
P-glycoprotein; glioblastoma multiforme; brain-blood barrier; doxorubicin
Online: 14 May 2018 (12:50:18 CEST)
ARTICLE
|
doi:10.20944/preprints202212.0135.v1
Subject:
Engineering,
Civil Engineering
Keywords:
Hydrodynamic model; marine and coastal tourism; analysis hierarchy process
Online: 7 December 2022 (14:47:31 CET)
ARTICLE
Subject:
Environmental And Earth Sciences,
Atmospheric Science And Meteorology
Keywords:
Ideal fluid; deep water; ice cover; moving cylinder; hydrodynamic load; added mass; wave resistance; damping coefficient
Online: 21 January 2021 (15:21:49 CET)
ARTICLE
|
doi:10.20944/preprints202312.0898.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
triazinyl phosphoramidate; amphiphilic oligonucleotides; self-assembly; human serum albumin; Ku antigen; PARP1; protein-oligonucleotide complexes
Online: 12 December 2023 (13:53:44 CET)
ARTICLE
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
(S)-Practolol; paracetamol; (S)-pindolol; (S)-carteolol; Candida antarctica Lipase B; chiral chromatography; dimer formation
Online: 4 March 2021 (08:34:02 CET)
ARTICLE
|
doi:10.20944/preprints202007.0056.v1
Subject:
Chemistry And Materials Science,
Materials Science And Technology
Keywords:
Aggregation-induced emission; quinones; fluorescence; TD-DFT; quantum yield
Online: 5 July 2020 (08:38:20 CEST)
BRIEF REPORT
|
doi:10.20944/preprints202001.0292.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
circadian rhythms; small molecules; luciferase reporters; period estimations
Online: 25 January 2020 (00:33:40 CET)