Search Results
38237 articles found
ARTICLE
|
doi:10.20944/preprints202311.0910.v1
Subject:
Medicine And Pharmacology,
Psychiatry And Mental Health
Keywords:
Antidepressants; Infertility; Males; Semen Quality; SSRIs
Online: 14 November 2023 (12:02:00 CET)
ARTICLE
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doi:10.20944/preprints202102.0589.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
serotonin transporter (SERT); thiadiazines; serotonin receptors 3 and 1A (5-HT3 and 5-HT1A); docking energy; binding affinity; binding mechanisms; electrophysiology in vivo
Online: 25 February 2021 (15:23:26 CET)
BRIEF REPORT
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doi:10.20944/preprints202403.0928.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
systemic sclerosis; pulmonary hypertension; Phosphodiesterase-5 inhibitors; endothelin receptor antagonist
Online: 15 March 2024 (13:15:50 CET)
REVIEW
|
doi:10.20944/preprints202408.1730.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Serotonin; Gut-Brain Interaction; Biomarker; Mood; Irritable Bowel Syndrome (IBS); Inflammatory Bowel Disease (IBD); Functional Dyspepsia (FD); Cancer; Gut Homeostasis
Online: 23 August 2024 (18:50:30 CEST)
REVIEW
|
doi:10.20944/preprints202402.0975.v1
Subject:
Medicine And Pharmacology,
Cardiac And Cardiovascular Systems
Keywords:
landiolol; atrial fibrillation; beta-blockers; perioperative tachyarrhythmias; cardiac surgery; arrhythmias
Online: 19 February 2024 (11:19:58 CET)
REVIEW
|
doi:10.20944/preprints202405.0059.v1
Subject:
Medicine And Pharmacology,
Dermatology
Keywords:
atopic dermatitis; calcineurin; NFAT; tacrolimus; pimecrolimus; cyclosporine
Online: 1 May 2024 (07:49:16 CEST)
ARTICLE
|
doi:10.20944/preprints202407.0037.v1
Subject:
Engineering,
Bioengineering
Keywords:
Serotonin, Fast Scan Cyclic Voltammetry, Boron Doped Diamond, Sensing, Neuroscience, Biomedical Engineering, Dopamine, Electrochemical Fouling, Neurotransmitter Detection, Microelectrodes
Online: 1 July 2024 (09:20:37 CEST)
ARTICLE
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doi:10.20944/preprints202402.1015.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Daridorexant; Insomnia; Orexin; Pharmacovigilance databases
Online: 19 February 2024 (16:14:12 CET)
REVIEW
|
doi:10.20944/preprints201808.0487.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
sex; anxiety disorders; 5-HT; tryptophan; immune system; inflammation
Online: 29 August 2018 (08:58:26 CEST)
REVIEW
|
doi:10.20944/preprints202208.0089.v1
Subject:
Social Sciences,
Behavior Sciences
Keywords:
Serotonin; Chemical imbalance theories of psychopathology; Circular causality; Biocultural psychopathology; Critical neuroscience
Online: 3 August 2022 (11:24:47 CEST)
ARTICLE
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doi:10.20944/preprints202405.0913.v1
Subject:
Medicine And Pharmacology,
Cardiac And Cardiovascular Systems
Keywords:
endothelin-receptor antagonist (ERA); bosentan; atorvastatin; atherosclerosis; plaque stability; matrix metalloproteinases
Online: 14 May 2024 (06:50:40 CEST)
REVIEW
|
doi:10.20944/preprints202404.0944.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Immune checkpoint inhibitor; ipilimumab; pembrolizumab
Online: 16 April 2024 (03:30:17 CEST)
COMMUNICATION
|
doi:10.20944/preprints202301.0334.v1
Subject:
Biology And Life Sciences,
Animal Science, Veterinary Science And Zoology
Keywords:
serotonin; pcpa; cystamine; dinophilida; invertebate models; aging; maternal serotonin; lifespan longevity
Online: 18 January 2023 (10:22:43 CET)
REVIEW
|
doi:10.20944/preprints202111.0529.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
TNFR2 Antagonist; TNFR2 Agonist; MDSCs; Treg; CD+Foxp3+
Online: 29 November 2021 (12:10:20 CET)
ARTICLE
|
doi:10.20944/preprints202407.1816.v1
Subject:
Biology And Life Sciences,
Neuroscience And Neurology
Keywords:
Agonist-antagonist myoneural interface; Electrical muscle stimulation; Muscle Reinnervation; Proprioception; Electromyograph; Targeted muscle reinnervation; Myoelectrical prosthesis; amputation; Peripheral nerve transfer; Compound action potential
Online: 23 July 2024 (18:00:18 CEST)
REVIEW
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doi:10.20944/preprints202405.0668.v3
Subject:
Biology And Life Sciences,
Neuroscience And Neurology
Keywords:
epilepsy; neuroinflammation; NLRP3 inflammasome; epileptogenesis; antiseizure medication; interleukin-1b; caspase-1; ASC
Online: 31 May 2024 (15:29:49 CEST)
ARTICLE
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doi:10.20944/preprints202104.0685.v1
Subject:
Social Sciences,
Psychology
Keywords:
gene-environment; serotonin transporter gene; 5HTTLPR; attachment; parent-infant interaction; parental bonding; maternal overprotection; close relationship; anxiety; avoidance
Online: 26 April 2021 (17:30:58 CEST)
REVIEW
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doi:10.20944/preprints202104.0676.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
RNA; Protamine; Transfection; Cancer Therapy; Vaccines
Online: 26 April 2021 (13:37:51 CEST)
REVIEW
|
doi:10.20944/preprints202201.0394.v1
Subject:
Social Sciences,
Psychology
Keywords:
parenting; 5HTTLPR; serotonin transporter; maternal sensitivity; polymorphism; gene X environment
Online: 26 January 2022 (12:19:45 CET)
REVIEW
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
apoptosis; antitumor; antimetastasis; anti-angiogenesis; NK-1 receptor; substance P; drug repositioning; Emend
Online: 31 August 2020 (10:11:13 CEST)
REVIEW
|
doi:10.20944/preprints202402.0872.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Immunotherapy; Immune checkpoint inhibitors; Rechallenge therapy; Resistance; NSCLC
Online: 16 February 2024 (11:34:11 CET)
REVIEW
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doi:10.20944/preprints202112.0174.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
Calcium channels; somatic exocytosis; serotonin; extrasynaptic release; leech
Online: 10 December 2021 (12:16:40 CET)
REVIEW
|
doi:10.20944/preprints201912.0096.v1
Subject:
Biology And Life Sciences,
Neuroscience And Neurology
Keywords:
brain connectivity; brain development; gut-brain axis; neurodevelopmental diseases; neuronal cytoarchitecture; neuroplasticity; regulatory T cells; serotonin (5-HT)
Online: 7 December 2019 (16:55:39 CET)
ARTICLE
|
doi:10.20944/preprints202403.1581.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
ASD-Phen1; STP1; ibudilast; bumetanide; phase 1b; EGG; NIH-TCB; SRS-2; ABC-C
Online: 26 March 2024 (10:20:29 CET)
ARTICLE
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
predator scent; aldosterone; corticosterone; adrenal gland; dorsal raphe nucleus (DRN); serotonin (5-HT); electrophysiology
Online: 15 July 2021 (10:40:31 CEST)
REVIEW
|
doi:10.20944/preprints202406.0880.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Dendritic cells; DC based cancer vaccine; Immune checkpoint inhibitors; Cancer Therapy; Combinatorial therapy
Online: 13 June 2024 (11:51:42 CEST)
ARTICLE
|
doi:10.20944/preprints201810.0746.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
aryl hydrocarbon receptor; polyphenols; inflammation; urolithin; AHR antagonist
Online: 31 October 2018 (10:08:59 CET)
REVIEW
|
doi:10.20944/preprints202408.0744.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
Peripheral T-cell lymphoma; Histone deacetylase (HDAC); HDAC inhibitor (HDACi); targeted therapy; epigenetic; DNA mutation; TET2; DNMT3A
Online: 12 August 2024 (05:07:04 CEST)
ARTICLE
|
doi:10.20944/preprints202403.0717.v1
Subject:
Biology And Life Sciences,
Animal Science, Veterinary Science And Zoology
Keywords:
Lumpy skin disease; DNA polymerase; potential inhibitors; phytocompounds; antiviral drug compounds; molecular docking
Online: 13 March 2024 (07:58:39 CET)
ARTICLE
|
doi:10.20944/preprints202112.0095.v1
Subject:
Medicine And Pharmacology,
Orthopedics And Sports Medicine
Keywords:
coactivation; agonist; strength; muscular performance; dynamic contraction; eccentric; concentric.
Online: 6 December 2021 (19:29:42 CET)
ARTICLE
|
doi:10.20944/preprints201801.0273.v2
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
antagonism; Bacillus velezensis; Penicillium roqueforti; silage; roquefortine C
Online: 1 March 2018 (14:24:15 CET)
ARTICLE
|
doi:10.20944/preprints202103.0309.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
CXCR4; EPI-X4; human serum albumin
Online: 11 March 2021 (10:55:07 CET)
REVIEW
|
doi:10.20944/preprints202205.0290.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
Cholesterol; PCSK9 inhibitors; HMG-CoA; LDL receptor; statins
Online: 23 May 2022 (10:01:24 CEST)
REVIEW
|
doi:10.20944/preprints202404.0091.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
menin; menin inhibitors; leukemia; KMT2A; NPM1
Online: 2 April 2024 (02:51:43 CEST)
ARTICLE
|
doi:10.20944/preprints202408.2012.v1
Subject:
Biology And Life Sciences,
Other
Keywords:
Herbacetin; (-)-Epicatechin; KATII inhibition; molecular docking; Molecular dynamic
Online: 28 August 2024 (09:37:19 CEST)
ARTICLE
|
doi:10.20944/preprints202404.1491.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
HIV-2; integrase strand transfer inhibitor (INSTIs); HIV; integrase; Lenacapavir; SARs-CoV-2
Online: 23 April 2024 (05:06:50 CEST)
ARTICLE
|
doi:10.20944/preprints202307.1008.v1
Subject:
Medicine And Pharmacology,
Surgery
Keywords:
Transtibial amputation; transfemoral amputation; agonist-antagonist myoneural interface; AMI; proprioception; neural interface; functional limb restoration; patient reported outcomes
Online: 14 July 2023 (13:29:21 CEST)
ARTICLE
|
doi:10.20944/preprints202407.0477.v1
Subject:
Medicine And Pharmacology,
Epidemiology And Infectious Diseases
Keywords:
DENV3; ZIKV; molecular docking; MD simulations; MM/GBSA; compound library; NS5; lycorine
Online: 5 July 2024 (12:04:10 CEST)
ARTICLE
|
doi:10.20944/preprints202407.1450.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Bladder cancer; STAT3 inhibitor; Apoptosis; Preclinical; 3D models
Online: 17 July 2024 (14:18:54 CEST)
COMMUNICATION
|
doi:10.20944/preprints202406.0315.v1
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
GLP-1 receptor agonist; liraglutide; serotonin; tryptophan; bile acids
Online: 10 June 2024 (12:22:04 CEST)
ARTICLE
|
doi:10.20944/preprints202409.0421.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Helicobacter pylori; antimicrobial resistance; narrow-spectrum antibiotic; antibacterial target; response regulator; HsrA; Campylobacter jejuni
Online: 5 September 2024 (10:22:25 CEST)
REVIEW
|
doi:10.20944/preprints202402.1049.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
malignant pleural mesothelioma; immune checkpoint inhibitor; orphan drug; good clinical practice; Pharmaceuticals and Medical Devices Agency
Online: 20 February 2024 (04:03:22 CET)
ARTICLE
|
doi:10.20944/preprints202406.2011.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
machine learning; prediction methods; cancer; ic50; r programming
Online: 29 June 2024 (05:59:44 CEST)
ARTICLE
|
doi:10.20944/preprints202402.1740.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Rheumatoid Arthritis, Anti-TNF, NRF2, Reverse Signaling, Biotherapy, Monoclonal Antibodies, Monocytes, Prediction.
Online: 29 February 2024 (14:46:26 CET)
REVIEW
|
doi:10.20944/preprints202312.0739.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Autoimmune diseases; Deficiency of Interluekin-1 Receptor Antagonist (DIRA); Anakinra; IL-1RA; IL-1RN
Online: 11 December 2023 (17:55:12 CET)
ARTICLE
|
doi:10.20944/preprints202403.1880.v1
Subject:
Public Health And Healthcare,
Other
Keywords:
Anti-interferon-γ autoantibodies; herpes zoster; monocyte chemoattractant protein-1; IFN-γ inducible protein-10; Janus kinas inhibitors; rheumatoid arthritis.
Online: 1 April 2024 (10:20:44 CEST)
ARTICLE
|
doi:10.20944/preprints202405.1741.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
Alzheimer’ s disease; vascular complications; monoclonal antibody therapy; Aducanumab; Lecanemab; epoxide of polyunsaturated fatty acid; soluble epoxide hydrolase inhibitor EC5026; EP4 inhibitor; monocyte/macrophage; amyloid-beta degradation
Online: 27 May 2024 (13:00:54 CEST)
ARTICLE
|
doi:10.20944/preprints201912.0374.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
alpha-fetoprotein; estrogens; selective estrogen receptor modulators; homology-based modeling; molecular docking; protein-ligand interaction; amino acid substitutions
Online: 29 December 2019 (08:08:23 CET)
REVIEW
|
doi:10.20944/preprints202401.0310.v1
Subject:
Medicine And Pharmacology,
Dentistry And Oral Surgery
Keywords:
inflammation; inflammasome; inhibitors of the inflammasome; nanomaterials; functionalized biomaterials; periodontitis; general pathology
Online: 4 January 2024 (09:25:17 CET)
REVIEW
|
doi:10.20944/preprints202306.0441.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
anti-lipoxygenase peptide; bioactivity; enzymatic hydrolysis; food peptide; food protein; inflammation; lipoxidase; lipoxygenase inhibitory activity.
Online: 6 June 2023 (10:11:09 CEST)
REVIEW
|
doi:10.20944/preprints202405.0573.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
Proton Pump Inhibitors (PPIs); Vonoprazan (VPZ); Intravenous infusion; Oral therapy; Bleeding peptic ulcers; Endoscopic therapy
Online: 9 May 2024 (09:15:54 CEST)
ARTICLE
|
doi:10.20944/preprints201609.0123.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
carbonic anhydrase; acetylcholinesterase; β-Lactam; 2-Azetidinone; enzyme inhibition; enzyme purification
Online: 30 September 2016 (05:38:45 CEST)
ARTICLE
|
doi:10.20944/preprints202405.0035.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Mycobacterial Polyketide Synthase; QSAR; Multiple Linear Regression; Docking; Molecular Dynamics Simulations
Online: 1 May 2024 (16:46:55 CEST)
ARTICLE
|
doi:10.20944/preprints202011.0456.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Intervertebral Disc; Renin-Angiotensin-System; Degeneration; Regeneration; Spine; Inflammation
Online: 17 November 2020 (14:48:38 CET)
ARTICLE
|
doi:10.20944/preprints202305.0004.v1
Subject:
Biology And Life Sciences,
Neuroscience And Neurology
Keywords:
neurodegeneration; traumatic brain injury; Zucker rat; Autoantibodies; serotonin 2A receptor
Online: 1 May 2023 (03:09:43 CEST)
ARTICLE
|
doi:10.20944/preprints202404.1152.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Tuberculosis; nitrobenzamides; DprE; mycobacteria
Online: 17 April 2024 (11:50:50 CEST)
REVIEW
|
doi:10.20944/preprints202204.0202.v1
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
Metabolic syndrome; SGLT2 inhibitors; Dapagliflozin; Empagliflozin; Canagliflozin; Translational modeling
Online: 21 April 2022 (10:12:04 CEST)
REVIEW
|
doi:10.20944/preprints202012.0167.v2
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Matrix metalloproteinase; MMPs; protease; TIMPs; exosite; small molecule inhibitors; monoclonal antibodies; proteomics; N-terminomics; TAILS
Online: 24 March 2021 (16:23:28 CET)
ARTICLE
|
doi:10.20944/preprints202405.0782.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Pancreatic cancer; pancreatic ductal adenocarcinoma; gemcitabine; growth hormone (GH); GH receptor (GHR); GHR antagonist; insulin-like growth factor 1 (IGF1); adjuvant; chemotherapy; chemoresistance
Online: 13 May 2024 (12:30:24 CEST)
ARTICLE
|
doi:10.20944/preprints202407.1916.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
cardiovascular disease; hepatic fibrosis; metabolic dysfunction-associated steatotic liver disease; sodium-glucose cotransporter 2 inhibitors; serum lipids
Online: 24 July 2024 (08:27:35 CEST)
REVIEW
|
doi:10.20944/preprints202401.0803.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
CYP enzymes; CYP3A4; flavonoid; inhibition; natural products
Online: 10 January 2024 (10:24:39 CET)
ARTICLE
|
doi:10.20944/preprints202307.0031.v1
Subject:
Chemistry And Materials Science,
Applied Chemistry
Keywords:
Ionic Liquids; Corrosion Inhibitors; Bio-based
Online: 4 July 2023 (02:23:59 CEST)
ARTICLE
|
doi:10.20944/preprints201710.0143.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
cheminformatics; docking simulation; drug repositioning; thiopurine; tyrosinase
Online: 22 October 2017 (14:03:13 CEST)
ARTICLE
|
doi:10.20944/preprints202406.0032.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
HIV-1; reverse transcriptase; polymerase; ribonuclease H; inhibitor; benzisothiazolone
Online: 3 June 2024 (07:56:06 CEST)
ARTICLE
|
doi:10.20944/preprints202208.0103.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Resveratrol; antioxidant metabolism; scavengome; biomimetic oxidation; bioactivity-guided isolation; NMR spectroscopy; xanthine oxidase
Online: 4 August 2022 (05:33:52 CEST)
ARTICLE
|
doi:10.20944/preprints202309.0253.v1
Subject:
Biology And Life Sciences,
Other
Keywords:
stess; chronic fatigue syndrome; depression; dysbiosis; serotonin/cortisol
Online: 5 September 2023 (07:52:50 CEST)
ARTICLE
|
doi:10.20944/preprints201701.0050.v1
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
Interleukin-1 receptor antagonist (IL-1Ra); Interleukin-4 (IL-4); Variable Number Tandem Repeat (VNTR); obesity; adiposity; Malaysia.
Online: 10 January 2017 (10:27:41 CET)
REVIEW
|
doi:10.20944/preprints202012.0419.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
immune checkpoint; lymphoid neoplasms; programmed death 1; cytotoxic T-lymphocyte antigen 4; monoclonal antibodies; combination therapies
Online: 17 December 2020 (08:10:05 CET)
ARTICLE
|
doi:10.20944/preprints202310.1571.v2
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Transketolase; malonylation; acetylation; sirtuin 5; oxythiamine; metformin; amprolium; thiamine; posttranslational modifications
Online: 10 November 2023 (12:03:31 CET)
REVIEW
|
doi:10.20944/preprints202406.0356.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
liver transplantation; hepatocellular carcinoma; Immune checkpoint inhibitors; allograft rejection
Online: 6 June 2024 (07:45:00 CEST)
ARTICLE
|
doi:10.20944/preprints202401.0776.v1
Subject:
Medicine And Pharmacology,
Urology And Nephrology
Keywords:
urothelial cancer; metastasis; prognosis; biomarker; pathway; autophagy
Online: 10 January 2024 (08:05:05 CET)
ARTICLE
|
doi:10.20944/preprints202111.0498.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
bortezomib; IL-13; IL-1Ra; IL-4; multiple myeloma; OS; PFS
Online: 26 November 2021 (10:31:50 CET)
REVIEW
|
doi:10.20944/preprints202404.0176.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
histone deacetylase inhibitors; radiosensitisation; heterochromatin; double strand break; DNA repair
Online: 2 April 2024 (10:09:33 CEST)
REVIEW
|
doi:10.20944/preprints202308.1413.v1
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
diabetes; cardiovascular; renal; SGLT1; SGLT2; therapy.
Online: 22 August 2023 (07:45:50 CEST)
REVIEW
|
doi:10.20944/preprints202307.1892.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Oncolytic virus; immune checkpoint inhibitors; immunotherapy
Online: 28 July 2023 (10:58:30 CEST)
ARTICLE
|
doi:10.20944/preprints202012.0383.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
meprin α; meprin β; zinc metalloproteinase; medicinal chemistry; probe development
Online: 15 December 2020 (12:56:31 CET)
ARTICLE
|
doi:10.20944/preprints202012.0354.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
meprin α; meprin β; zinc metalloproteinase; uHTS
Online: 14 December 2020 (16:36:57 CET)
HYPOTHESIS
|
doi:10.20944/preprints202004.0151.v2
Online: 22 April 2020 (09:46:54 CEST)
ARTICLE
|
doi:10.20944/preprints202408.1642.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
allogeneic hematopoietic stem cell transplantation; chronic myeloid leukaemia; tyrosine kinase inhibitors; imatinib; dasatinib; nilotinib
Online: 22 August 2024 (16:30:22 CEST)
ARTICLE
|
doi:10.20944/preprints202101.0319.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
thromboxane A2 and prostaglandin H2 receptor (TPR) antagonist; ONO-8809; renal disorders; salt-overload; stroke-prone spontaneously hypertensive rat (SHRSP); hypertension; oxidative stress
Online: 18 January 2021 (11:32:11 CET)
REVIEW
|
doi:10.20944/preprints202004.0224.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
substance P,; NK-1R,; AML,; Aprepitant,; anti-leukemic,; apoptosis,; non-solid tumor
Online: 14 April 2020 (15:19:45 CEST)
REVIEW
|
doi:10.20944/preprints202311.0295.v1
Subject:
Medicine And Pharmacology,
Cardiac And Cardiovascular Systems
Keywords:
Atrial fibrillation, SGLT2 inhibitors, cardiovascular outcomes, hemodynamic effects, AF risk reduction
Online: 6 November 2023 (08:13:49 CET)
ARTICLE
|
doi:10.20944/preprints202404.0785.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
enteroviruses, coxsackievirus, leucoverdazyls, antioxidant, antiviral, 2C protein
Online: 11 April 2024 (09:22:02 CEST)
REVIEW
|
doi:10.20944/preprints202401.1697.v1
Subject:
Medicine And Pharmacology,
Cardiac And Cardiovascular Systems
Keywords:
DOAC; FXIa; mAbs; ASO; drug-drug interactions
Online: 23 January 2024 (12:31:04 CET)
REVIEW
|
doi:10.20944/preprints202305.1761.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
checkpoint inhibitors; colitis; immune-related adverse events; enterocolitis; diarrhea
Online: 25 May 2023 (08:03:37 CEST)
ARTICLE
|
doi:10.20944/preprints202302.0423.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
B-cell; autoimmune disease; drug repurposing
Online: 24 February 2023 (09:11:37 CET)
REVIEW
|
doi:10.20944/preprints202402.1535.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
DNA polymerase I; Polymerase θ ; reverse transcriptase; homologous recombination; antibiotics; apicoplast
Online: 27 February 2024 (12:29:29 CET)
REVIEW
|
doi:10.20944/preprints202304.0516.v1
Subject:
Medicine And Pharmacology,
Internal Medicine
Keywords:
SGLT-2 Inhibitors; Inflammasome; NLRP3; reno-protective effects; Cardio-protective effects; neuro-protective effects.
Online: 18 April 2023 (10:33:39 CEST)
ARTICLE
|
doi:10.20944/preprints202211.0356.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Focal adhesion kinase; 3D-QSAR; Molecular Dynamics; MM-PB/GBSA; Free energy perturbation
Online: 18 November 2022 (10:13:00 CET)
ARTICLE
|
doi:10.20944/preprints202108.0001.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Antitumoral drug; Choline kinase inhibition; Choline uptake
Online: 2 August 2021 (08:42:22 CEST)
ARTICLE
|
doi:10.20944/preprints202408.1759.v1
Subject:
Biology And Life Sciences,
Neuroscience And Neurology
Keywords:
HIV; ferritin heavy-chain; ferritin light-chain; ferroptosis; lipid peroxidation; iron; oxidative stress; neurocognitive impairment; neurocognitive domains
Online: 24 August 2024 (00:22:41 CEST)
REVIEW
|
doi:10.20944/preprints202309.1651.v1
Subject:
Biology And Life Sciences,
Endocrinology And Metabolism
Keywords:
cyclic AMP; cyclic PIP; insulin resistance; prostaglandylinositol cyclic phosphate; protein phosphorylation; protein kinase A; protein ser/thr phosphatase; type 2 diabetes
Online: 25 September 2023 (11:05:29 CEST)
ARTICLE
|
doi:10.20944/preprints202312.1461.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
indirect comparison; Shiny method; reconstructed individual patient data; disease free survival; renal cell carcinoma; adjuvant setting
Online: 20 December 2023 (09:30:07 CET)
ARTICLE
|
doi:10.20944/preprints201703.0116.v1
Subject:
Biology And Life Sciences,
Animal Science, Veterinary Science And Zoology
Keywords:
In vivo; Alpha-glucosidase; Alpha-amylase; hyperglycemia
Online: 16 March 2017 (09:35:36 CET)
ARTICLE
|
doi:10.20944/preprints202408.1282.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Cataract; CRYGD; Molecular docking; Molecular dynamics; Crystallin; Protein aggregation
Online: 19 August 2024 (09:15:05 CEST)
ARTICLE
|
doi:10.20944/preprints202004.0240.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
COVID19; 2019-nCov, 3CLpro inhbitors
Online: 15 April 2020 (10:00:52 CEST)
ARTICLE
|
doi:10.20944/preprints202002.0047.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
2019-nCoV; therapeutic strategies; drug; ACE2
Online: 4 February 2020 (10:59:25 CET)
REVIEW
|
doi:10.20944/preprints201909.0140.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
hepatocellular carcinoma; immune checkpoint inhibitors; HCC; pembrolizumab; nivolumab; immune microenvironment; targeted therapies
Online: 14 September 2019 (18:37:29 CEST)
REVIEW
|
doi:10.20944/preprints201805.0145.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
carbonic anhydrase, enzyme inhibition, metalloenzymes, amino acid, glaucoma, tumors
Online: 9 May 2018 (13:55:15 CEST)
ARTICLE
|
doi:10.20944/preprints202311.0483.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
MRONJ; CDK4/6 inhibitors; metastatic breast cancer; oral epidemiology
Online: 8 November 2023 (08:42:55 CET)