Search Results
38686 articles found
ARTICLE
|
doi:10.20944/preprints202403.0552.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
S. sclerotiorum; Pathogenicity; Histone methylation; Mycotoxins; Stress.
Online: 11 March 2024 (09:56:54 CET)
REVIEW
|
doi:10.20944/preprints202111.0164.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
SETMAR; Metnase; H3K36me2; Hsmar1; non-homologous end joining repair; NHEJ; transposase; transposable elements; histone; methyltransferase
Online: 9 November 2021 (11:30:21 CET)
REVIEW
|
doi:10.20944/preprints202312.1587.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Cancer; Molecular Oncology; Oncogenes; NSD3; NSD3S
Online: 21 December 2023 (09:21:20 CET)
ARTICLE
|
doi:10.20944/preprints202406.1311.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
Coronavirus; SARS-CoV-2; MERS-CoV; 3CLPro; antivirals; protease inhibitors
Online: 19 June 2024 (05:53:52 CEST)
ARTICLE
|
doi:10.20944/preprints202208.0159.v1
Subject:
Biology And Life Sciences,
Endocrinology And Metabolism
Keywords:
metabolomics; NMR; PEMT; knockout; aging; mice; liver; intestine; white/brown adipose tissue
Online: 8 August 2022 (13:36:04 CEST)
REVIEW
|
doi:10.20944/preprints202409.1669.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
eIF4A; mTORC2-Akt pathway; β-catenin pathway; JNK pathway; paclitaxel; doxorubicin; fluorouracil; platinum-containing drug; IGF1R/IR inhibitor
Online: 23 September 2024 (11:53:36 CEST)
ARTICLE
|
doi:10.20944/preprints201701.0040.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Sarcocystis neurona; EPM; docking; apicomplexans; phylogeny; homology modeling
Online: 9 January 2017 (05:19:32 CET)
ARTICLE
|
doi:10.20944/preprints202408.1498.v1
Subject:
Biology And Life Sciences,
Horticulture
Keywords:
Cauliflower; Bax inhibitor-1; Expression pattern; BobBIL4; Abiotic stress
Online: 21 August 2024 (00:12:19 CEST)
ARTICLE
|
doi:10.20944/preprints202305.2047.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
CDC20; BIOMARKER; KMT5A; p53; prostate cancer
Online: 30 May 2023 (05:03:54 CEST)
ARTICLE
|
doi:10.20944/preprints202405.1076.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
soybean; Glycine max; Antinutritional factors; Bowman-Birk inhibitor; CRISPR-Cas9
Online: 16 May 2024 (17:23:37 CEST)
ARTICLE
|
doi:10.20944/preprints202409.0006.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
Melanoma metastasis; Ulcerative Colitis; Crohn's Disease; Rheumatoid arthritis; Integrated bioinformatics analysis; Virtual screening; Molecular docking; Molecular dynamic simulation
Online: 2 September 2024 (13:12:50 CEST)
ARTICLE
|
doi:10.20944/preprints202410.0041.v1
Subject:
Biochemistry And Molecular Biology,
Biology And Life Sciences
Keywords:
NNMT; ccRCC; biomarker
Online: 1 October 2024 (10:44:43 CEST)
ARTICLE
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
h. pylori; restriction modification system; virulence; il-8; apoptosis
Online: 1 November 2019 (12:52:39 CET)
REVIEW
|
doi:10.20944/preprints202308.0651.v1
Subject:
Biology And Life Sciences,
Other
Keywords:
cancer; adhesion; metastasis; inhibition; therapeutic approaches; targeted therapies
Online: 9 August 2023 (02:48:16 CEST)
REVIEW
|
doi:10.20944/preprints202402.0835.v3
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Hypertension; calcium channel blocker; combination therapy; thiazide diuretics; Renin-angiotensin-aldosterone system inhibitor
Online: 25 July 2024 (00:11:59 CEST)
ARTICLE
|
doi:10.20944/preprints202404.1491.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
HIV-2; integrase strand transfer inhibitor (INSTIs); HIV; integrase; Lenacapavir; SARs-CoV-2
Online: 23 April 2024 (05:06:50 CEST)
ARTICLE
|
doi:10.20944/preprints201610.0016.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
molecular dynamics simulation; virtual screening; molecular docking; prostate cancer; caveolin-1
Online: 7 October 2016 (12:09:06 CEST)
ARTICLE
|
doi:10.20944/preprints202406.0791.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
p-gp; p-glycoprotein; AU1; BPTF inhibitor; triple negative breast cancer; efflux pump; multidrug resistance; multidrug resistance pump; breast cancer
Online: 12 June 2024 (11:58:34 CEST)
ARTICLE
|
doi:10.20944/preprints202407.1888.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Keywords: Coronavirus; 3CL protease; Drug target for Coronavirus; SARS-CoV
Online: 24 July 2024 (12:36:54 CEST)
ARTICLE
|
doi:10.20944/preprints201708.0021.v1
Subject:
Chemistry And Materials Science,
Surfaces, Coatings And Films
Keywords:
3-((2-chlorobenzylidene)amino)coumarin; corrosion inhibitor; damage reduction
Online: 7 August 2017 (10:51:42 CEST)
ARTICLE
|
doi:10.20944/preprints202401.0325.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Menaquinone; inhibitor; Mycobacterium tuberculosis; MIC; IC50
Online: 4 January 2024 (09:49:21 CET)
SHORT NOTE
|
doi:10.20944/preprints201707.0096.v1
Subject:
Chemistry And Materials Science,
Surfaces, Coatings And Films
Keywords:
corrosion inhibitor; coumarin; resonance
Online: 31 July 2017 (16:37:19 CEST)
CONCEPT PAPER
|
doi:10.20944/preprints202004.0213.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
covid-19; rlmE MTase; new drug target; corona diagnosis; corona pandemic
Online: 13 April 2020 (12:33:22 CEST)
ARTICLE
|
doi:10.20944/preprints202407.2417.v1
Subject:
Biology And Life Sciences,
Endocrinology And Metabolism
Keywords:
ACAT1/SOAT1; nanoparticle; F1251; F26; cholesterol; cholesteryl ester; DSPE-PEG; phosphatidylcholine; neurodegenerative diseases; Alzheimer’s disease
Online: 30 July 2024 (07:35:59 CEST)
TECHNICAL NOTE
|
doi:10.20944/preprints201706.0085.v1
Subject:
Engineering,
Civil Engineering
Keywords:
finite element modeling; electrochemical chloride extraction (ECE); electrical injection of corrosion inhibitor (EICI); rebar corrosion; repair mortar
Online: 19 June 2017 (13:40:09 CEST)
ARTICLE
|
doi:10.20944/preprints202403.0251.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Neurobastoma; Radionuclide therapy; Apoptosis; Somatostatin analog; Radiosensitization; Combination therapy
Online: 5 March 2024 (13:05:37 CET)
ARTICLE
|
doi:10.20944/preprints202405.1856.v1
Subject:
Environmental And Earth Sciences,
Soil Science
Keywords:
soil N turnover; straw application; nitrification inhibitor; 15N labeling; 15N recovery; 15N retention; nitrogen use efficiency; Mollisol
Online: 29 May 2024 (04:15:24 CEST)
REVIEW
|
doi:10.20944/preprints202405.2008.v2
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
immune checkpoint inhibitor; aging; cellular senescence; immune-related adverse events
Online: 10 June 2024 (04:21:20 CEST)
ARTICLE
|
doi:10.20944/preprints202408.1683.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Immunotherapy; Celiac Disease; Enterocolitis; CTLA-4; HLA-DQ2; PD-L1; PD-1; Adverse Effects; Gluten-Free Diet
Online: 23 August 2024 (12:21:14 CEST)
REVIEW
|
doi:10.20944/preprints202105.0140.v1
Subject:
Engineering,
Automotive Engineering
Keywords:
Adsorption; Scale Inhibitors; Fine sands; Colloids; Reservoir
Online: 7 May 2021 (10:42:36 CEST)
ARTICLE
|
doi:10.20944/preprints202403.1581.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
ASD-Phen1; STP1; ibudilast; bumetanide; phase 1b; EGG; NIH-TCB; SRS-2; ABC-C
Online: 26 March 2024 (10:20:29 CET)
ARTICLE
|
doi:10.20944/preprints202312.0493.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
pathogens; IspE inhibitor; carboline, synthesis; minimum inhibitory concentration
Online: 7 December 2023 (16:54:59 CET)
REVIEW
|
doi:10.20944/preprints202401.1900.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Tunicamycin; Nanoparticle; Immunotherapy; Glycosylation; Drug resistance; Multidrug therapy; cancer
Online: 26 January 2024 (11:39:36 CET)
ARTICLE
|
doi:10.20944/preprints202306.1841.v1
Subject:
Biology And Life Sciences,
Animal Science, Veterinary Science And Zoology
Keywords:
Piceatannol; Pseudorabies virus; Antiviral activity; in vivo; in vitro
Online: 27 June 2023 (03:08:19 CEST)
ARTICLE
|
doi:10.20944/preprints202205.0001.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
ovarian cancer; ALDH1A1; cancer stem cells; senescence; chemotherapy resistance
Online: 2 May 2022 (09:39:22 CEST)
ARTICLE
|
doi:10.20944/preprints202102.0520.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Meprin B; Meprin beta; metalloproteinase; astacin; hydroxamate; SAR (structure activity relationship); MWT-S-270
Online: 23 February 2021 (14:27:53 CET)
ARTICLE
|
doi:10.20944/preprints202012.0414.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
galantamine; curcumin; in vivo AChE inhibition; acute toxicity in mice; antioxidant activity; malondialdehide levels; glutathione levels; brain homogenate; complete blood count; biochemical serum parameters
Online: 16 December 2020 (13:45:10 CET)
REVIEW
|
doi:10.20944/preprints201909.0120.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Lysophosphatidic acid; Autotaxin; inhibitor; allosteric; orthosteric; lipid chaperone; signalling, GPCR
Online: 11 September 2019 (13:18:21 CEST)
REVIEW
|
doi:10.20944/preprints201807.0254.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
endocrine disruptor, environmental health sciences, gene-environment, inhibitor of differentiation, neurocognitive disorders
Online: 14 July 2018 (23:30:36 CEST)
CASE REPORT
|
doi:10.20944/preprints202404.0157.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
autoimmune encephalitis; checkpoint inhibitor; melanoma; pembrolizumab; adverse event
Online: 2 April 2024 (16:18:10 CEST)
ARTICLE
|
doi:10.20944/preprints201809.0525.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
hepatitis E virus; innate immunity; interferon response; JAK/STAT pathway; zoonosis; emerging pathogen
Online: 27 September 2018 (03:34:49 CEST)
ARTICLE
|
doi:10.20944/preprints202409.0112.v1
Subject:
Medicine And Pharmacology,
Dermatology
Keywords:
Diabetic wound; Human β -defensin-2; Matrix metalloproteinase-9; Protein kinase C-β II; Protein-protein docking; Molecular dynamics simulation studies
Online: 2 September 2024 (13:35:48 CEST)
ARTICLE
|
doi:10.20944/preprints202308.1350.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Imidazole; Imidazole derivative; Sirtuins; NSCLC; Epigenetics
Online: 18 August 2023 (09:04:18 CEST)
ARTICLE
|
doi:10.20944/preprints202308.0569.v1
Subject:
Medicine And Pharmacology,
Dermatology
Keywords:
Keratinocytes; alpha-mangostin; TRPV3; skin inflammation; dermatitis
Online: 8 August 2023 (03:42:33 CEST)
ARTICLE
|
doi:10.20944/preprints202009.0523.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
Anticancer; Tubulin; HSP27; Nimesulide; SKOV3; SKBR3
Online: 22 September 2020 (15:19:02 CEST)
ARTICLE
|
doi:10.20944/preprints201901.0086.v1
Subject:
Business, Economics And Management,
Finance
Keywords:
Quinoxaline Analogs, Synthesis, Thymidine phosphorylase inhibition, Molecular docking
Online: 9 January 2019 (13:23:49 CET)
ARTICLE
|
doi:10.20944/preprints202407.0432.v1
Subject:
Medicine And Pharmacology,
Internal Medicine
Keywords:
ventilator-associated pneumonia; biomarkers; pediatric intensive care unit; critically-ill children; ventilator-associated pneumonia; biomarkers; pediatric intensive care unit; critically-ill children
Online: 4 July 2024 (11:00:29 CEST)
ARTICLE
|
doi:10.20944/preprints202304.0601.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
FTSJ1; methyltransferase; tRNA; readthrough; stop codon mutation; small molecules; docking; molecular dynamics; MM-GBSA
Online: 20 April 2023 (03:21:07 CEST)
ARTICLE
|
doi:10.20944/preprints202312.0574.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
DOCK program; GOLD program; Grb14; insulin receptor (IR); structure-based drug screening (SBDS)
Online: 8 December 2023 (08:24:15 CET)
COMMUNICATION
|
doi:10.20944/preprints202305.0704.v2
Subject:
Chemistry And Materials Science,
Other
Keywords:
protein-protein interaction inhibitor; rule of five; rule of four; QEPPI; molecular generation; virtual chemical library
Online: 30 June 2023 (08:50:24 CEST)
ARTICLE
|
doi:10.20944/preprints202211.0068.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Pancreatic cancer; metabolism; metformin; NAD; NAMPT
Online: 3 November 2022 (03:38:59 CET)
ARTICLE
|
doi:10.20944/preprints201804.0374.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
STAT3 as a drug target; cyclic STAT3 decoy; oligodeoxynucleotide inhibitor; head and neck cancer
Online: 29 April 2018 (10:10:00 CEST)
ARTICLE
|
doi:10.20944/preprints202309.2155.v1
Subject:
Biology And Life Sciences,
Animal Science, Veterinary Science And Zoology
Keywords:
beraprost; feline; chronic kidney disease; aldosterone; NOS
Online: 30 September 2023 (05:18:01 CEST)
ARTICLE
|
doi:10.20944/preprints202302.0250.v1
Subject:
Medicine And Pharmacology,
Other
Keywords:
AI drug discovery; mTOR; rapalog; C. elegans; cancer; longevity
Online: 15 February 2023 (02:42:57 CET)
ARTICLE
|
doi:10.20944/preprints202105.0600.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
heparan sulfate; glycosaminoglycan; carbohydrate biosynthesis; azido sugar; small molecule inhibitor
Online: 25 May 2021 (10:17:59 CEST)
ARTICLE
|
doi:10.20944/preprints202103.0655.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
mitochondria; Ca2+ handling; heart failure; CaMKII; cardiomyocyte hypertrophy
Online: 26 March 2021 (10:41:00 CET)
ARTICLE
|
doi:10.20944/preprints202403.1760.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
JAK-inhibitor; baricitinib; rheumatoid arthritis; real-word data; persistence; adherence; safety; unmet needs.
Online: 28 March 2024 (10:30:28 CET)
ARTICLE
|
doi:10.20944/preprints202308.1349.v1
Subject:
Biology And Life Sciences,
Neuroscience And Neurology
Keywords:
α-Synuclein preformed fibrils (PFF); cytotoxicity; Reactive Oxygen Species (ROS); oxidative stress; and protein aggregation
Online: 18 August 2023 (10:55:57 CEST)
ARTICLE
|
doi:10.20944/preprints202308.1071.v1
Subject:
Biology And Life Sciences,
Neuroscience And Neurology
Keywords:
Alzheimer’s disease; DPTIP; hydroxyl PAMAM dendrimer; D-DPTIP; extracellular vesicles; neutral sphingomyelinase 2; tau
Online: 15 August 2023 (09:01:43 CEST)
ARTICLE
|
doi:10.20944/preprints201807.0131.v1
Subject:
Medicine And Pharmacology,
Ophthalmology
Keywords:
pigmentary glaucoma; ROCK kinase inhibitor; RKI-1447; trabecular meshwork; phagocytosis; cytoskeleton
Online: 9 July 2018 (11:27:28 CEST)
ARTICLE
|
doi:10.20944/preprints201802.0026.v1
Subject:
Medicine And Pharmacology,
Ophthalmology
Keywords:
pig eye perfusion model; pigmentary glaucoma; ocular hypertension; ocular hypotension; phagocytosis; rho-kinase inhibitor
Online: 5 February 2018 (03:39:57 CET)
ARTICLE
|
doi:10.20944/preprints202104.0170.v1
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
abdominal subcutaneous adipocytes; angiotensinogen; nuclear factor-kappa B; lipopolysaccharide; tumor necrosis factor-alpha
Online: 6 April 2021 (11:28:00 CEST)
ARTICLE
|
doi:10.20944/preprints202406.2035.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Cannabidiol; MAPK; EGFR; Ras/Raf; colorectal cancer
Online: 2 July 2024 (09:19:32 CEST)
ARTICLE
|
doi:10.20944/preprints202311.0910.v1
Subject:
Medicine And Pharmacology,
Psychiatry And Mental Health
Keywords:
Antidepressants; Infertility; Males; Semen Quality; SSRIs
Online: 14 November 2023 (12:02:00 CET)
ARTICLE
|
doi:10.20944/preprints202308.0231.v1
Subject:
Public Health And Healthcare,
Public Health And Health Services
Keywords:
G protein-coupled receptors, Protease Activated Receptor2; Allosteric modulator; 1-piperidinepropionic acid; Molecular Dynamics.
Online: 2 August 2023 (13:20:19 CEST)
COMMUNICATION
|
doi:10.20944/preprints202306.0701.v1
Subject:
Medicine And Pharmacology,
Urology And Nephrology
Keywords:
Iron isomaltoside; NF-kappaBeta; dehydroxymethyepoxyquinmicin (DHMEQ); mesothelial cells
Online: 9 June 2023 (10:37:47 CEST)
ARTICLE
|
doi:10.20944/preprints202205.0393.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
poxviruses; protein kinase R; evolution; translational regulation; eIF2
Online: 30 May 2022 (10:42:41 CEST)
ARTICLE
|
doi:10.20944/preprints202204.0183.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
resistant TNBC; intra-tumoral heterogeneity; breast cancer relapse; breast cancer epigenome; me-tastasis prevention; intrinsic resistance of cancer; tumor adaptability; targeting resistant cancer
Online: 20 April 2022 (04:16:31 CEST)
ARTICLE
|
doi:10.20944/preprints202203.0405.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
α-amylase inhibitors; diabetes; hemi-pyocyanin; marine discards; microbial conversion
Online: 31 March 2022 (10:47:24 CEST)
ARTICLE
|
doi:10.20944/preprints202108.0100.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
PF-543; ceramide; SPHK; SPT; ceramide synthases; sphingolipid; metabolism; LC-MS/MS.
Online: 4 August 2021 (08:32:59 CEST)
ARTICLE
|
doi:10.20944/preprints202408.0507.v1
Subject:
Engineering,
Civil Engineering
Keywords:
admixture; concrete; sodium benzoate; corrosion inhibitor; limestone fillers; mechanical resistance; time
Online: 7 August 2024 (14:01:28 CEST)
ARTICLE
|
doi:10.20944/preprints202211.0137.v1
Subject:
Medicine And Pharmacology,
Dermatology
Keywords:
Mushroom tyrosinase; Melanogenesis; Tyrosinase inhibitor; Multi-spectroscopic techniques; Natural compounds; tyrosinase inhibitor
Online: 8 November 2022 (02:23:25 CET)
REVIEW
|
doi:10.20944/preprints202105.0285.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
PP2A; LB100; nervous system; tumor biology; brain tumor; preclinical; clinical trial
Online: 13 May 2021 (11:32:51 CEST)
ARTICLE
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
propolis; pro- and anti-inflammatory cytokines; LPS stimulation; bone marrow derived macrophages; metabolomics
Online: 14 September 2020 (00:36:37 CEST)
REVIEW
|
doi:10.20944/preprints201810.0732.v1
Subject:
Social Sciences,
Behavior Sciences
Keywords:
depression; estrogenic endocrine disruptor; environmental factor; inhibitor of differentiation; mental disorder
Online: 31 October 2018 (04:51:16 CET)
ARTICLE
|
doi:10.20944/preprints202306.1963.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Glioblastoma Multiform (GBM); Cancer Stem Cella (CSC); Molecular Dynamics Simulation; In-silico; Phytochemical Screening; FOXM1; ADMET
Online: 28 June 2023 (08:23:27 CEST)
REVIEW
|
doi:10.20944/preprints202306.1955.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
breast cancer; CDK4/6 inhibitors; estrogen receptor; therapeutic resistance
Online: 28 June 2023 (07:39:44 CEST)
ARTICLE
|
doi:10.20944/preprints202306.0548.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
non-alcoholic steatohepatitis; hepatocellular carcinoma; farnesyltransferase inhibitor; hypoxia-inducible factor-1α; anti-inflammatory response; nuclear factor-κB; transforming growth factor-β; Warburg effect; reactive oxygen species; interleukin-6
Online: 7 June 2023 (12:05:28 CEST)
ARTICLE
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Oleuropein; colon cancer; activated macrophages; chronic inflammation; inducible nitric oxide synthetase (iNOS); cyclooxygenase-2 (COX-2); nitric oxide (NO)
Online: 2 August 2021 (12:04:58 CEST)
ARTICLE
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
3,4-dimethoxy-β-nitrostyrene derivatives; antimicrobial agent; PTP1B; molecular docking
Online: 20 July 2020 (11:31:48 CEST)
COMMUNICATION
|
doi:10.20944/preprints202409.0083.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
Dengue; docking simulations; Autodock Vina; Amentoflavone
Online: 2 September 2024 (09:49:45 CEST)
ARTICLE
|
doi:10.20944/preprints202305.0538.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
Aging; Betaine; dBHMT; Drosophila; dSAMTOR; dTORC1; Kinase; Methionine; SAM
Online: 8 May 2023 (12:06:37 CEST)
CASE REPORT
|
doi:10.20944/preprints202206.0266.v1
Subject:
Medicine And Pharmacology,
Pathology And Pathobiology
Keywords:
PARP inhibitor; angiogenesis; immune suppression; recurrent ovarian cancer
Online: 20 June 2022 (10:02:09 CEST)
ARTICLE
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
K-Ras; Hsp90; Cdc37; nanoclustering; cancer; drug development
Online: 31 March 2021 (15:30:27 CEST)
ARTICLE
|
doi:10.20944/preprints201810.0133.v2
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
aging; angiotensin-converting enzyme inhibitors; nutrient metabolism; genetic background; nutritional stress
Online: 29 October 2018 (10:33:59 CET)
ARTICLE
|
doi:10.20944/preprints202407.1116.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Hepatitis C virus; MD Simulations; Covalent inhibitor; Drug resistance; Pharmacophore-based virtual screening
Online: 16 July 2024 (04:54:08 CEST)
ARTICLE
|
doi:10.20944/preprints202106.0297.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Trueperella pyogenes; TatD DNases; luteolin; DNA hydrolysis; molecular modeling; SPR
Online: 10 June 2021 (14:13:37 CEST)
ARTICLE
|
doi:10.20944/preprints202308.1001.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
Brass; Corrosion; Inhibition efficiency; ESBB
Online: 14 August 2023 (09:39:15 CEST)
ARTICLE
|
doi:10.20944/preprints202308.0291.v1
Subject:
Biology And Life Sciences,
Agricultural Science And Agronomy
Keywords:
hypocotyl growth; neurotransmitter; root growth; skototropism; γ-aminobutyric acid
Online: 3 August 2023 (07:21:57 CEST)
ARTICLE
|
doi:10.20944/preprints202010.0477.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Exportin-1; Eriodictyol; Juglans mandshurica; Non-small cell lung cancer
Online: 23 October 2020 (10:19:32 CEST)
ARTICLE
|
doi:10.20944/preprints202305.1403.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Alzheimer’s Disease; Tauopathy; Cell penetrating peptide; Polyarginine; TAT; Liposomes; Nanoparticles; Tau pathology; Tau aggregation inhibitor; Endocytosis
Online: 19 May 2023 (08:06:10 CEST)
CONCEPT PAPER
|
doi:10.20944/preprints202004.0282.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
SARS-CoV-2; Penicillamine; spike protein; docking
Online: 16 April 2020 (15:44:39 CEST)
ARTICLE
|
doi:10.20944/preprints202004.0084.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
in silico repositioning; dual inhibitor; Covid-19; 3CLpro; PLpro; remdesivir
Online: 7 April 2020 (10:44:11 CEST)
ARTICLE
|
doi:10.20944/preprints201808.0146.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
histone deacetylase inhibitor, MHY2256, p53, apoptosis, autophagy, Ishikawa, endometrial cancer
Online: 7 August 2018 (14:37:46 CEST)
REVIEW
|
doi:10.20944/preprints202306.1788.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Meningioma; Cabozantinib; VEGF; Targeted treatment Cabozantinib; METs; VEGFR2; Inhibitors; Angiogen-esis; Oncology
Online: 26 June 2023 (10:57:00 CEST)
ARTICLE
|
doi:10.20944/preprints202305.0217.v1
Subject:
Chemistry And Materials Science,
Materials Science And Technology
Keywords:
mild Steel; corrosion rate; dioscorea spp; NaOH; NaCl; H2SO4
Online: 4 May 2023 (07:44:22 CEST)
ARTICLE
|
doi:10.20944/preprints202106.0115.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
triterpenoids; Acacia stem bark; polypharmacology; protein kinase inhibitors
Online: 3 June 2021 (13:04:47 CEST)
ARTICLE
|
doi:10.20944/preprints201909.0124.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Heat shock factor (HSF-1) knockdown; heat shock proteins 70 and 27; radiosensitization; Hsp90 inhibitor NVP-AUY922; homologous recombination (HR)
Online: 11 September 2019 (13:37:00 CEST)
REVIEW
|
doi:10.20944/preprints201907.0286.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
HIV-1 Gag; Gag inhibitors; Protease; Protease inhibitors; drug resistance mutations; drug design
Online: 25 July 2019 (10:05:03 CEST)
ARTICLE
|
doi:10.20944/preprints201811.0247.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Inonotus Obliquus, Melanogenesis, B16F10, Tyrosinase, MITF
Online: 9 November 2018 (13:36:36 CET)