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DRUG: Drospirenone and estradiol
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Entry
D12497 Mixture Drug
Name
Drospirenone and estradiol;
Angeliq (TN)
Product
ANGELIQ (Bayer HealthCare Pharmaceuticals)
Component
Drospirenone [DR:
D03917
], (Estradiol [DR:
D00105
] | Estradiol hemihydrate [DR:
D07918
])
Class
Metabolizing enzyme substrate
DG01633
CYP3A/CYP3A4 substrate
DG02913
CYP3A4 substrate
Remark
Product:
D12497<US>
Efficacy
Contraceptive
Comment
Drospirenone is primarily metabolized by CYP3A4.
Metabolism
Enzyme: CYP3A4 [HSA:
1576
]
Interaction
DDI search
Brite
Drug groups [BR:
br08330
]
Metabolizing enzyme substrate
DG01633 CYP3A/CYP3A4 substrate
DG02913 CYP3A4 substrate
D12497 Drospirenone and estradiol
Drug metabolizing enzymes and transporters [
br08309.html
]
Drug metabolizing enzymes
D12497
BRITE hierarchy
Other DBs
PubChem:
497620910
LinkDB
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