Search Results
38495 articles found
ARTICLE
|
doi:10.20944/preprints202311.1799.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
usnic acid derivatives; TDP1 inhibitors; anticancer therapy; topotecan
Online: 28 November 2023 (10:06:47 CET)
ARTICLE
|
doi:10.20944/preprints202312.0002.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
tyrosyl-DNA phosphodiesterase 1; topoisomerase 1; HEK293A; transcriptome; TDP1 knockout
Online: 1 December 2023 (04:53:45 CET)
REVIEW
|
doi:10.20944/preprints202405.0059.v1
Subject:
Medicine And Pharmacology,
Dermatology
Keywords:
atopic dermatitis; calcineurin; NFAT; tacrolimus; pimecrolimus; cyclosporine
Online: 1 May 2024 (07:49:16 CEST)
REVIEW
|
doi:10.20944/preprints202404.0944.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Immune checkpoint inhibitor; ipilimumab; pembrolizumab
Online: 16 April 2024 (03:30:17 CEST)
REVIEW
|
doi:10.20944/preprints202405.0668.v3
Subject:
Biology And Life Sciences,
Neuroscience And Neurology
Keywords:
epilepsy; neuroinflammation; NLRP3 inflammasome; epileptogenesis; antiseizure medication; interleukin-1b; caspase-1; ASC
Online: 31 May 2024 (15:29:49 CEST)
REVIEW
|
doi:10.20944/preprints202402.0872.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Immunotherapy; Immune checkpoint inhibitors; Rechallenge therapy; Resistance; NSCLC
Online: 16 February 2024 (11:34:11 CET)
REVIEW
|
doi:10.20944/preprints202406.0880.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Dendritic cells; DC based cancer vaccine; Immune checkpoint inhibitors; Cancer Therapy; Combinatorial therapy
Online: 13 June 2024 (11:51:42 CEST)
REVIEW
|
doi:10.20944/preprints202408.0744.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
Peripheral T-cell lymphoma; Histone deacetylase (HDAC); HDAC inhibitor (HDACi); targeted therapy; epigenetic; DNA mutation; TET2; DNMT3A
Online: 12 August 2024 (05:07:04 CEST)
ARTICLE
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doi:10.20944/preprints202403.0717.v1
Subject:
Biology And Life Sciences,
Animal Science, Veterinary Science And Zoology
Keywords:
Lumpy skin disease; DNA polymerase; potential inhibitors; phytocompounds; antiviral drug compounds; molecular docking
Online: 13 March 2024 (07:58:39 CET)
REVIEW
|
doi:10.20944/preprints202205.0290.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
Cholesterol; PCSK9 inhibitors; HMG-CoA; LDL receptor; statins
Online: 23 May 2022 (10:01:24 CEST)
REVIEW
|
doi:10.20944/preprints202404.0091.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
menin; menin inhibitors; leukemia; KMT2A; NPM1
Online: 2 April 2024 (02:51:43 CEST)
ARTICLE
|
doi:10.20944/preprints202408.2012.v1
Subject:
Biology And Life Sciences,
Other
Keywords:
Herbacetin; (-)-Epicatechin; KATII inhibition; molecular docking; Molecular dynamic
Online: 28 August 2024 (09:37:19 CEST)
ARTICLE
|
doi:10.20944/preprints202404.1491.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
HIV-2; integrase strand transfer inhibitor (INSTIs); HIV; integrase; Lenacapavir; SARs-CoV-2
Online: 23 April 2024 (05:06:50 CEST)
ARTICLE
|
doi:10.20944/preprints202407.0477.v1
Subject:
Medicine And Pharmacology,
Epidemiology And Infectious Diseases
Keywords:
DENV3; ZIKV; molecular docking; MD simulations; MM/GBSA; compound library; NS5; lycorine
Online: 5 July 2024 (12:04:10 CEST)
ARTICLE
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doi:10.20944/preprints202407.1450.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Bladder cancer; STAT3 inhibitor; Apoptosis; Preclinical; 3D models
Online: 17 July 2024 (14:18:54 CEST)
ARTICLE
|
doi:10.20944/preprints202409.0421.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Helicobacter pylori; antimicrobial resistance; narrow-spectrum antibiotic; antibacterial target; response regulator; HsrA; Campylobacter jejuni
Online: 5 September 2024 (10:22:25 CEST)
REVIEW
|
doi:10.20944/preprints202402.1049.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
malignant pleural mesothelioma; immune checkpoint inhibitor; orphan drug; good clinical practice; Pharmaceuticals and Medical Devices Agency
Online: 20 February 2024 (04:03:22 CET)
ARTICLE
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doi:10.20944/preprints202406.2011.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
machine learning; prediction methods; cancer; ic50; r programming
Online: 29 June 2024 (05:59:44 CEST)
ARTICLE
|
doi:10.20944/preprints202402.1740.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Rheumatoid Arthritis, Anti-TNF, NRF2, Reverse Signaling, Biotherapy, Monoclonal Antibodies, Monocytes, Prediction.
Online: 29 February 2024 (14:46:26 CET)
ARTICLE
|
doi:10.20944/preprints202403.1880.v1
Subject:
Public Health And Healthcare,
Other
Keywords:
Anti-interferon-γ autoantibodies; herpes zoster; monocyte chemoattractant protein-1; IFN-γ inducible protein-10; Janus kinas inhibitors; rheumatoid arthritis.
Online: 1 April 2024 (10:20:44 CEST)
ARTICLE
|
doi:10.20944/preprints202405.1741.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
Alzheimer’ s disease; vascular complications; monoclonal antibody therapy; Aducanumab; Lecanemab; epoxide of polyunsaturated fatty acid; soluble epoxide hydrolase inhibitor EC5026; EP4 inhibitor; monocyte/macrophage; amyloid-beta degradation
Online: 27 May 2024 (13:00:54 CEST)
BRIEF REPORT
|
doi:10.20944/preprints202403.0928.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
systemic sclerosis; pulmonary hypertension; Phosphodiesterase-5 inhibitors; endothelin receptor antagonist
Online: 15 March 2024 (13:15:50 CET)
REVIEW
|
doi:10.20944/preprints202401.0310.v1
Subject:
Medicine And Pharmacology,
Dentistry And Oral Surgery
Keywords:
inflammation; inflammasome; inhibitors of the inflammasome; nanomaterials; functionalized biomaterials; periodontitis; general pathology
Online: 4 January 2024 (09:25:17 CET)
REVIEW
|
doi:10.20944/preprints202306.0441.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
anti-lipoxygenase peptide; bioactivity; enzymatic hydrolysis; food peptide; food protein; inflammation; lipoxidase; lipoxygenase inhibitory activity.
Online: 6 June 2023 (10:11:09 CEST)
REVIEW
|
doi:10.20944/preprints202405.0573.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
Proton Pump Inhibitors (PPIs); Vonoprazan (VPZ); Intravenous infusion; Oral therapy; Bleeding peptic ulcers; Endoscopic therapy
Online: 9 May 2024 (09:15:54 CEST)
ARTICLE
|
doi:10.20944/preprints201609.0123.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
carbonic anhydrase; acetylcholinesterase; β-Lactam; 2-Azetidinone; enzyme inhibition; enzyme purification
Online: 30 September 2016 (05:38:45 CEST)
ARTICLE
|
doi:10.20944/preprints202405.0035.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Mycobacterial Polyketide Synthase; QSAR; Multiple Linear Regression; Docking; Molecular Dynamics Simulations
Online: 1 May 2024 (16:46:55 CEST)
REVIEW
|
doi:10.20944/preprints202204.0202.v1
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
Metabolic syndrome; SGLT2 inhibitors; Dapagliflozin; Empagliflozin; Canagliflozin; Translational modeling
Online: 21 April 2022 (10:12:04 CEST)
REVIEW
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doi:10.20944/preprints202012.0167.v2
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Matrix metalloproteinase; MMPs; protease; TIMPs; exosite; small molecule inhibitors; monoclonal antibodies; proteomics; N-terminomics; TAILS
Online: 24 March 2021 (16:23:28 CET)
ARTICLE
|
doi:10.20944/preprints202404.1152.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Tuberculosis; nitrobenzamides; DprE; mycobacteria
Online: 17 April 2024 (11:50:50 CEST)
ARTICLE
|
doi:10.20944/preprints202407.1916.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
cardiovascular disease; hepatic fibrosis; metabolic dysfunction-associated steatotic liver disease; sodium-glucose cotransporter 2 inhibitors; serum lipids
Online: 24 July 2024 (08:27:35 CEST)
REVIEW
|
doi:10.20944/preprints202401.0803.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
CYP enzymes; CYP3A4; flavonoid; inhibition; natural products
Online: 10 January 2024 (10:24:39 CET)
ARTICLE
|
doi:10.20944/preprints202307.0031.v1
Subject:
Chemistry And Materials Science,
Applied Chemistry
Keywords:
Ionic Liquids; Corrosion Inhibitors; Bio-based
Online: 4 July 2023 (02:23:59 CEST)
ARTICLE
|
doi:10.20944/preprints201710.0143.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
cheminformatics; docking simulation; drug repositioning; thiopurine; tyrosinase
Online: 22 October 2017 (14:03:13 CEST)
ARTICLE
|
doi:10.20944/preprints202406.0032.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
HIV-1; reverse transcriptase; polymerase; ribonuclease H; inhibitor; benzisothiazolone
Online: 3 June 2024 (07:56:06 CEST)
ARTICLE
|
doi:10.20944/preprints202208.0103.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Resveratrol; antioxidant metabolism; scavengome; biomimetic oxidation; bioactivity-guided isolation; NMR spectroscopy; xanthine oxidase
Online: 4 August 2022 (05:33:52 CEST)
REVIEW
|
doi:10.20944/preprints202012.0419.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
immune checkpoint; lymphoid neoplasms; programmed death 1; cytotoxic T-lymphocyte antigen 4; monoclonal antibodies; combination therapies
Online: 17 December 2020 (08:10:05 CET)
ARTICLE
|
doi:10.20944/preprints202310.1571.v2
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Transketolase; malonylation; acetylation; sirtuin 5; oxythiamine; metformin; amprolium; thiamine; posttranslational modifications
Online: 10 November 2023 (12:03:31 CET)
REVIEW
|
doi:10.20944/preprints202406.0356.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
liver transplantation; hepatocellular carcinoma; Immune checkpoint inhibitors; allograft rejection
Online: 6 June 2024 (07:45:00 CEST)
REVIEW
|
doi:10.20944/preprints202404.0176.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
histone deacetylase inhibitors; radiosensitisation; heterochromatin; double strand break; DNA repair
Online: 2 April 2024 (10:09:33 CEST)
REVIEW
|
doi:10.20944/preprints202308.1413.v1
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
diabetes; cardiovascular; renal; SGLT1; SGLT2; therapy.
Online: 22 August 2023 (07:45:50 CEST)
REVIEW
|
doi:10.20944/preprints202307.1892.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Oncolytic virus; immune checkpoint inhibitors; immunotherapy
Online: 28 July 2023 (10:58:30 CEST)
ARTICLE
|
doi:10.20944/preprints202012.0383.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
meprin α; meprin β; zinc metalloproteinase; medicinal chemistry; probe development
Online: 15 December 2020 (12:56:31 CET)
ARTICLE
|
doi:10.20944/preprints202012.0354.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
meprin α; meprin β; zinc metalloproteinase; uHTS
Online: 14 December 2020 (16:36:57 CET)
HYPOTHESIS
|
doi:10.20944/preprints202004.0151.v2
Online: 22 April 2020 (09:46:54 CEST)
ARTICLE
|
doi:10.20944/preprints202408.1642.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
allogeneic hematopoietic stem cell transplantation; chronic myeloid leukaemia; tyrosine kinase inhibitors; imatinib; dasatinib; nilotinib
Online: 22 August 2024 (16:30:22 CEST)
REVIEW
|
doi:10.20944/preprints202311.0295.v1
Subject:
Medicine And Pharmacology,
Cardiac And Cardiovascular Systems
Keywords:
Atrial fibrillation, SGLT2 inhibitors, cardiovascular outcomes, hemodynamic effects, AF risk reduction
Online: 6 November 2023 (08:13:49 CET)
ARTICLE
|
doi:10.20944/preprints202404.0785.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
enteroviruses, coxsackievirus, leucoverdazyls, antioxidant, antiviral, 2C protein
Online: 11 April 2024 (09:22:02 CEST)
REVIEW
|
doi:10.20944/preprints202401.1697.v1
Subject:
Medicine And Pharmacology,
Cardiac And Cardiovascular Systems
Keywords:
DOAC; FXIa; mAbs; ASO; drug-drug interactions
Online: 23 January 2024 (12:31:04 CET)
REVIEW
|
doi:10.20944/preprints202305.1761.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
checkpoint inhibitors; colitis; immune-related adverse events; enterocolitis; diarrhea
Online: 25 May 2023 (08:03:37 CEST)
ARTICLE
|
doi:10.20944/preprints202302.0423.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
B-cell; autoimmune disease; drug repurposing
Online: 24 February 2023 (09:11:37 CET)
REVIEW
|
doi:10.20944/preprints202402.1535.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
DNA polymerase I; Polymerase θ ; reverse transcriptase; homologous recombination; antibiotics; apicoplast
Online: 27 February 2024 (12:29:29 CET)
REVIEW
|
doi:10.20944/preprints202304.0516.v1
Subject:
Medicine And Pharmacology,
Internal Medicine
Keywords:
SGLT-2 Inhibitors; Inflammasome; NLRP3; reno-protective effects; Cardio-protective effects; neuro-protective effects.
Online: 18 April 2023 (10:33:39 CEST)
ARTICLE
|
doi:10.20944/preprints202211.0356.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Focal adhesion kinase; 3D-QSAR; Molecular Dynamics; MM-PB/GBSA; Free energy perturbation
Online: 18 November 2022 (10:13:00 CET)
ARTICLE
|
doi:10.20944/preprints202108.0001.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Antitumoral drug; Choline kinase inhibition; Choline uptake
Online: 2 August 2021 (08:42:22 CEST)
ARTICLE
|
doi:10.20944/preprints202408.1759.v1
Subject:
Biology And Life Sciences,
Neuroscience And Neurology
Keywords:
HIV; ferritin heavy-chain; ferritin light-chain; ferroptosis; lipid peroxidation; iron; oxidative stress; neurocognitive impairment; neurocognitive domains
Online: 24 August 2024 (00:22:41 CEST)
ARTICLE
|
doi:10.20944/preprints202312.1461.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
indirect comparison; Shiny method; reconstructed individual patient data; disease free survival; renal cell carcinoma; adjuvant setting
Online: 20 December 2023 (09:30:07 CET)
ARTICLE
|
doi:10.20944/preprints201703.0116.v1
Subject:
Biology And Life Sciences,
Animal Science, Veterinary Science And Zoology
Keywords:
In vivo; Alpha-glucosidase; Alpha-amylase; hyperglycemia
Online: 16 March 2017 (09:35:36 CET)
ARTICLE
|
doi:10.20944/preprints202408.1282.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Cataract; CRYGD; Molecular docking; Molecular dynamics; Crystallin; Protein aggregation
Online: 19 August 2024 (09:15:05 CEST)
ARTICLE
|
doi:10.20944/preprints202004.0240.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
COVID19; 2019-nCov, 3CLpro inhbitors
Online: 15 April 2020 (10:00:52 CEST)
ARTICLE
|
doi:10.20944/preprints202002.0047.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
2019-nCoV; therapeutic strategies; drug; ACE2
Online: 4 February 2020 (10:59:25 CET)
REVIEW
|
doi:10.20944/preprints201909.0140.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
hepatocellular carcinoma; immune checkpoint inhibitors; HCC; pembrolizumab; nivolumab; immune microenvironment; targeted therapies
Online: 14 September 2019 (18:37:29 CEST)
REVIEW
|
doi:10.20944/preprints201805.0145.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
carbonic anhydrase, enzyme inhibition, metalloenzymes, amino acid, glaucoma, tumors
Online: 9 May 2018 (13:55:15 CEST)
ARTICLE
|
doi:10.20944/preprints202311.0483.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
MRONJ; CDK4/6 inhibitors; metastatic breast cancer; oral epidemiology
Online: 8 November 2023 (08:42:55 CET)
ARTICLE
|
doi:10.20944/preprints202307.2034.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Bcl-2; Anti-apoptotic protein; Indole; Cancer drug discovery
Online: 28 July 2023 (14:36:37 CEST)
ARTICLE
|
doi:10.20944/preprints202107.0270.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
drug design; falcipain; malaria; peptidomimetics; Plasmodium falciparum; virtual screening; pharmacophore.
Online: 12 July 2021 (14:48:13 CEST)
REVIEW
|
doi:10.20944/preprints202106.0158.v1
Online: 7 June 2021 (09:29:06 CEST)
ARTICLE
|
doi:10.20944/preprints201811.0330.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
hyperpigmentation; tyrosinase inhibitors; 3-(2,4-dihydroxyphenyl)propionic acid; structure-activity relationship study; B16-F10 cellular melanogenesis inhibition
Online: 14 November 2018 (09:59:45 CET)
ARTICLE
|
doi:10.20944/preprints201801.0213.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
bichalcones; sirtuin inhibitors; virtual screening
Online: 23 January 2018 (09:12:43 CET)
ARTICLE
|
doi:10.20944/preprints202307.1251.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
ascorbic acid; pharmacologic ascorbate; pancreatic cancer; epigenetics; DNA methyltransferase (DNMT); ten-eleven translocation (TET) methylcytosine dioxygenase
Online: 18 July 2023 (13:51:14 CEST)
REVIEW
|
doi:10.20944/preprints202405.0992.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
proteases; viruses; respiratory proteases; protease inhibitors; SARS-CoV-2
Online: 15 May 2024 (10:29:30 CEST)
ARTICLE
|
doi:10.20944/preprints202308.0468.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
dasatinib; imatinib; nilotibin; ponatinib; children; therapeutic drug monitoring; sex and gender pharmacology; personalized medicine.
Online: 7 August 2023 (11:53:12 CEST)
REVIEW
|
doi:10.20944/preprints202305.1151.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
fusion proteins; inhibitor; therapeutic; cancer
Online: 16 May 2023 (10:32:09 CEST)
REVIEW
|
doi:10.20944/preprints202211.0448.v1
Subject:
Medicine And Pharmacology,
Pulmonary And Respiratory Medicine
Keywords:
alpha-1-antitrypsin (AAT); neutrophil elastase (NE); NETosis, PAD4, ARDS, COPD; neutrophils; COVID-19; TMPRSS2.
Online: 24 November 2022 (02:50:25 CET)
ARTICLE
|
doi:10.20944/preprints201911.0375.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
synthesis; 2-mercaptabezimidazole; sulfonamide; molecular docking study; α-amylase; sa
Online: 29 November 2019 (10:28:22 CET)
ARTICLE
|
doi:10.20944/preprints201801.0196.v1
Subject:
Medicine And Pharmacology,
Urology And Nephrology
Keywords:
comorbid diseases; erectile dysfunction; penile duplex doppler ultrasound; penile pathology; phosphodiesterase type 5 inhibitors
Online: 22 January 2018 (09:03:17 CET)
ARTICLE
|
doi:10.20944/preprints202403.1095.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
KRAS inhibitor; metastasis; colorectal cancer; machine learning; meta analysis
Online: 21 March 2024 (03:50:20 CET)
ARTICLE
|
doi:10.20944/preprints202308.0290.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
RNA-binding protein; human antigen R (HuR); high-throughput virtual screening; small molecule inhibitors; RNA pulldown assay
Online: 3 August 2023 (10:11:15 CEST)
ARTICLE
|
doi:10.20944/preprints202307.0433.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
PCNA; p15; FRET; inhibitor screening; ATLD2; disease; variant; stability; aggregation
Online: 6 July 2023 (11:53:02 CEST)
REVIEW
|
doi:10.20944/preprints202306.0956.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
NSCLC,; Immunotherapy; Immune Checkpoint Inhibitors; Special populations
Online: 13 June 2023 (16:01:04 CEST)
ARTICLE
|
doi:10.20944/preprints202306.0109.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
triple negative breast cancer; MCAK/KIF2C; aneuploidy; chromosomal instability; drug discovery
Online: 1 June 2023 (15:47:29 CEST)
REVIEW
|
doi:10.20944/preprints202204.0065.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
COVID-19; Main protease; Mpro; inhibitors
Online: 8 April 2022 (03:01:37 CEST)
REVIEW
|
doi:10.20944/preprints201806.0056.v1
Subject:
Medicine And Pharmacology,
Pathology And Pathobiology
Keywords:
mTOR; mTORC1; mTORC2; rapamycin; rapalogues; rapalogs; mTOR inhibitors; senescence; ageing; aging; cancer; neurodegeneration; immunosenescence; senolytics; biomarkers
Online: 5 June 2018 (09:49:19 CEST)
ARTICLE
|
doi:10.20944/preprints202307.1626.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Proton pump inhibitors; Clopidogrel; Stroke; Myocardial infarction
Online: 25 July 2023 (07:26:31 CEST)
ARTICLE
|
doi:10.20944/preprints202307.0765.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
4-amino-7-chloroquinoline; 1,3,4-oxadiazole; anthranilic acid; synthesis; quorum sensing; anti-biofilm; P. aeruginosa; PQS
Online: 12 July 2023 (21:25:14 CEST)
REVIEW
|
doi:10.20944/preprints202306.0614.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
frailty, comorbidities, Crohn's disease, ulcerative colitis, infections, malignancies
Online: 8 June 2023 (09:30:13 CEST)
ARTICLE
|
doi:10.20944/preprints202205.0097.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
KV1.3; potassium ion channels; antiproliferative activity; apoptosis; anticancer drugs
Online: 9 May 2022 (03:35:09 CEST)
ARTICLE
|
doi:10.20944/preprints202402.1288.v2
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
SGLT2 Inhibitors; Empagliflozin; Renal fibrosis; Connective tissue growth factor; Epithelial-mesenchymal transition
Online: 23 February 2024 (13:25:01 CET)
REVIEW
|
doi:10.20944/preprints202409.1354.v1
Subject:
Medicine And Pharmacology,
Cardiac And Cardiovascular Systems
Keywords:
superoxide; SGLT2 inhibitors; GLP-1 agonists; cardiorenal syndrome; diuretic resistance; heart failure
Online: 18 September 2024 (11:37:54 CEST)
ARTICLE
|
doi:10.20944/preprints202312.1702.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
vascular prosthesis; AEBSF; puromycin; Staphylococcus aureus; FTIR analysis
Online: 22 December 2023 (08:03:49 CET)
REVIEW
|
doi:10.20944/preprints202306.1426.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Trypanosomatids; squalene synthase; farnesyl diphosphate synthase; target-based approach; neglected tropical diseases.
Online: 20 June 2023 (10:27:48 CEST)
ARTICLE
|
doi:10.20944/preprints202209.0218.v1
Subject:
Chemistry And Materials Science,
Theoretical Chemistry
Keywords:
Scutellaria baicalensis; phytochemicals; glioblastoma multiforme; in silico
Online: 15 September 2022 (03:55:58 CEST)
ARTICLE
|
doi:10.20944/preprints202201.0243.v1
Subject:
Chemistry And Materials Science,
Food Chemistry
Keywords:
aqueous micellar system; trypsin inhibitor; isoflavone extraction; non-ionic surfactant; multifactorial optimization
Online: 17 January 2022 (16:01:53 CET)
REVIEW
|
doi:10.20944/preprints202112.0282.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Acalabrutinib; Bruton’s tyrosine kinase; BTK; CLL; Covalent inhibitors; COVID-19; Ibrutinib; Non-covalent inhibitors; Fenebrutinib; MK1026; Pirtobrutinib; Spebrutinib; Tirabrutinib; Zanubrutinib
Online: 16 December 2021 (16:13:54 CET)
ARTICLE
|
doi:10.20944/preprints201909.0130.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Synthesis; triazinoindole; thiosemicarbazide; alpha-glucosidase; molecular docking study; SAR
Online: 13 September 2019 (10:54:30 CEST)
ARTICLE
|
doi:10.20944/preprints201710.0200.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
4-Thiazolidinones; ORAC assay; Metalloproteinase-9; Docking study; Keratinocytes cultures; Nuclear factor -kB.
Online: 31 October 2017 (16:36:16 CET)
ARTICLE
|
doi:10.20944/preprints201709.0070.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Coumarin; Mycobacterium tuberculosis; Cholinesterase inhibitor; Monoamine oxidase B inhibitor; Structure activity relationship; Albumin binding, Neuroprotection
Online: 15 September 2017 (17:34:38 CEST)
REVIEW
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
hyperoxaluria; oxalate; inhibitor; small molecule drug; glycolate oxidase; lactate dehydrogenase; liver selective distribution
Online: 31 December 2020 (08:59:47 CET)
COMMUNICATION
|
doi:10.20944/preprints202004.0146.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Coronavirus Disease 2019; SARS-CoV-2; main protease; molecular docking-based virtual screening
Online: 9 April 2020 (09:34:45 CEST)
REVIEW
|
doi:10.20944/preprints201807.0116.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
chemical space; chemoinformatics; data mining; databases; DNMT inhibitors; drug discovery; epi-informatics; molecular modeling; similarity searching; virtual screening
Online: 6 July 2018 (10:04:44 CEST)