Search Results
36946 articles found
ARTICLE
|
doi:10.20944/preprints202302.0423.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
B-cell; autoimmune disease; drug repurposing
Online: 24 February 2023 (09:11:37 CET)
ARTICLE
|
doi:10.20944/preprints202308.0468.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
dasatinib; imatinib; nilotibin; ponatinib; children; therapeutic drug monitoring; sex and gender pharmacology; personalized medicine.
Online: 7 August 2023 (11:53:12 CEST)
ARTICLE
|
doi:10.20944/preprints202209.0218.v1
Subject:
Chemistry And Materials Science,
Theoretical Chemistry
Keywords:
Scutellaria baicalensis; phytochemicals; glioblastoma multiforme; in silico
Online: 15 September 2022 (03:55:58 CEST)
ARTICLE
Subject:
Computer Science And Mathematics,
Mathematical And Computational Biology
Keywords:
c-src-tyrosine kinase; QSAR; molecular descriptors; virtual screening; drug discovery; cancer; molecular docking
Online: 25 October 2019 (11:21:43 CEST)
ARTICLE
|
doi:10.20944/preprints202312.1461.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
indirect comparison; Shiny method; reconstructed individual patient data; disease free survival; renal cell carcinoma; adjuvant setting
Online: 20 December 2023 (09:30:07 CET)
ARTICLE
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doi:10.20944/preprints202305.1022.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
N-methyl piperazine; Dubermatinib; In vitro metabolites; Cyano adducts; GSH conjugate; Xe-nosite reactivity model
Online: 15 May 2023 (10:28:28 CEST)
REVIEW
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
EGFR-mutated non-small cell lung cancer; EGFR-TKI; intrinsic resistance; resistance mechanisms
Online: 22 April 2019 (11:08:42 CEST)
REVIEW
|
doi:10.20944/preprints202107.0353.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Lung cancer; Adjuvant treatment; Non-small-cell lung carcinoma (NSCLC); Epidermal growth factor receptor (EGFR); Tyrosine kinase inhibitor (TKI)
Online: 15 July 2021 (10:16:30 CEST)
REVIEW
|
doi:10.20944/preprints202305.1789.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
PTK6; Colorectal cancer; Tyrosine Kinase Inhibitors
Online: 25 May 2023 (09:52:24 CEST)
ARTICLE
|
doi:10.20944/preprints202408.1642.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
allogeneic hematopoietic stem cell transplantation; chronic myeloid leukaemia; tyrosine kinase inhibitors; imatinib; dasatinib; nilotinib
Online: 22 August 2024 (16:30:22 CEST)
ARTICLE
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doi:10.20944/preprints202211.0356.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Focal adhesion kinase; 3D-QSAR; Molecular Dynamics; MM-PB/GBSA; Free energy perturbation
Online: 18 November 2022 (10:13:00 CET)
ARTICLE
|
doi:10.20944/preprints202108.0001.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Antitumoral drug; Choline kinase inhibition; Choline uptake
Online: 2 August 2021 (08:42:22 CEST)
REVIEW
|
doi:10.20944/preprints202306.1788.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Meningioma; Cabozantinib; VEGF; Targeted treatment Cabozantinib; METs; VEGFR2; Inhibitors; Angiogen-esis; Oncology
Online: 26 June 2023 (10:57:00 CEST)
ARTICLE
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doi:10.20944/preprints202403.1880.v1
Subject:
Public Health And Healthcare,
Other
Keywords:
Anti-interferon-γ autoantibodies; herpes zoster; monocyte chemoattractant protein-1; IFN-γ inducible protein-10; Janus kinas inhibitors; rheumatoid arthritis.
Online: 1 April 2024 (10:20:44 CEST)
ARTICLE
|
doi:10.20944/preprints202407.2128.v1
Subject:
Medicine And Pharmacology,
Urology And Nephrology
Keywords:
metastatic renal cell carcinoma; tyrosine kinase inhibitor sunitinib; nomogram; cancer-specific survival; prognosis; treatment response
Online: 26 July 2024 (06:23:32 CEST)
REVIEW
|
doi:10.20944/preprints202307.0990.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
Bruton's tyrosine kinase (BTK); cognitive disorders; multiple sclerosis (MS); Neuroinflammation; immune system
Online: 14 July 2023 (13:24:12 CEST)
ARTICLE
|
doi:10.20944/preprints201908.0177.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
chronic myeloid leukemia; tyrosine kinase inhibitor; adverse drug event; quality of life; second-generation tyrosine kinase inhibitor; nilotinib
Online: 16 August 2019 (08:09:07 CEST)
ARTICLE
|
doi:10.20944/preprints202107.0195.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
Loop-mediated isothermal amplification; AXL over expression; core-shell beads assay
Online: 8 July 2021 (10:57:31 CEST)
REVIEW
|
doi:10.20944/preprints202112.0282.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Acalabrutinib; Bruton’s tyrosine kinase; BTK; CLL; Covalent inhibitors; COVID-19; Ibrutinib; Non-covalent inhibitors; Fenebrutinib; MK1026; Pirtobrutinib; Spebrutinib; Tirabrutinib; Zanubrutinib
Online: 16 December 2021 (16:13:54 CET)
ARTICLE
|
doi:10.20944/preprints202403.1433.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
FLT3 Inhibitors; Ligand-based Drug Design; Computer-Aided Drug Design; QSAR Modeling; AML Treatment
Online: 25 March 2024 (08:47:40 CET)
ARTICLE
|
doi:10.20944/preprints202305.1252.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
iPSCs; HSCs; RET; Hematopoietic differentiation; CD34
Online: 17 May 2023 (13:49:58 CEST)
ARTICLE
|
doi:10.20944/preprints201908.0238.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
aurora kinase A; molecular docking; DFT; MD simulation
Online: 23 August 2019 (05:01:40 CEST)
ARTICLE
|
doi:10.20944/preprints202105.0638.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
18F-FDG PET/CT; contrast-enhanced CT; melanoma; metastases; tyrosine kinase inhibitors; Immune checkpoint inhibitors; follow-up; therapy monitoring
Online: 26 May 2021 (13:14:06 CEST)
ARTICLE
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
18F-FDG PET/CT; contrast-enhanced CT; melanoma; metastases; tyrosine kinase inhibitors; Immune checkpoint inhibitors; follow-up; therapy monitoring
Online: 25 January 2021 (15:01:17 CET)
REVIEW
|
doi:10.20944/preprints202307.2046.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
CADD; SBDD; LBDD; kinase; small molecule kinase inhibitors
Online: 31 July 2023 (03:05:42 CEST)
ARTICLE
|
doi:10.20944/preprints202104.0174.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Phosphodiesterase (PDE); natural products; inhibitors; Protein Kinase; selectivity; fluorescence polarization
Online: 6 April 2021 (12:07:58 CEST)
ARTICLE
|
doi:10.20944/preprints202404.0651.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Cholangiocyte – primary liver cancer – selumetinib – AZD6244 – MK2206 – intrahepatic cholangiocarcinoma
Online: 9 April 2024 (10:56:59 CEST)
ARTICLE
|
doi:10.20944/preprints201709.0082.v1
Subject:
Medicine And Pharmacology,
Dietetics And Nutrition
Keywords:
tyrosine; dose-response; aging; working memory; plasma amino acids; catecholamines; dopamine
Online: 18 September 2017 (15:48:07 CEST)
REVIEW
|
doi:10.20944/preprints202405.0059.v1
Subject:
Medicine And Pharmacology,
Dermatology
Keywords:
atopic dermatitis; calcineurin; NFAT; tacrolimus; pimecrolimus; cyclosporine
Online: 1 May 2024 (07:49:16 CEST)
ARTICLE
|
doi:10.20944/preprints202408.1876.v1
Subject:
Biology And Life Sciences,
Aging
Keywords:
life span; aging; Drosophila; rapamycin; TOR inhibition
Online: 26 August 2024 (17:13:59 CEST)
ARTICLE
|
doi:10.20944/preprints202403.1229.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
PTPRE; miR631; retinoblastoma; CAM assay; etoposide; chemoresistance; tumorigenesis
Online: 20 March 2024 (13:13:44 CET)
ARTICLE
|
doi:10.20944/preprints202312.0595.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
chronic myeloid leukemia; tyrosine kinase inhibitor; very elderly; safety; efficacy; outcome; dose optimization
Online: 8 December 2023 (10:26:16 CET)
ARTICLE
|
doi:10.20944/preprints202402.0640.v1
Subject:
Computer Science And Mathematics,
Mathematical And Computational Biology
Keywords:
Lung adenocarcinoma; EGFR TKI; precision oncology; in silico; computational oncology
Online: 12 February 2024 (10:57:20 CET)
REVIEW
|
doi:10.20944/preprints202203.0274.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
dopamine; locus coeruleus; melanin; neuromelanin; norepinephrine; Parkinson’s disease; substan-tia nigra; tyrosinase; tyrosine hydroxylase
Online: 21 March 2022 (05:14:47 CET)
REVIEW
|
doi:10.20944/preprints202404.0944.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Immune checkpoint inhibitor; ipilimumab; pembrolizumab
Online: 16 April 2024 (03:30:17 CEST)
REVIEW
|
doi:10.20944/preprints202405.0668.v3
Subject:
Biology And Life Sciences,
Neuroscience And Neurology
Keywords:
epilepsy; neuroinflammation; NLRP3 inflammasome; epileptogenesis; antiseizure medication; interleukin-1b; caspase-1; ASC
Online: 31 May 2024 (15:29:49 CEST)
ARTICLE
|
doi:10.20944/preprints202407.1375.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
CacyBP/SIP; ERK1/2; p38; seminoma; testis
Online: 17 July 2024 (04:56:33 CEST)
ARTICLE
|
doi:10.20944/preprints202406.0034.v1
Subject:
Biology And Life Sciences,
Neuroscience And Neurology
Keywords:
voltage-gated sodium channels; fibroblast growth factors; split luciferase assay; kinase inhibitors
Online: 3 June 2024 (08:07:35 CEST)
ARTICLE
|
doi:10.20944/preprints202311.0018.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
protein tyrosine phosphatases; polymerase and histidinol phosphatases; Cap8C; Wzb; metal ion activation; thermophilic enzymes
Online: 1 November 2023 (09:49:36 CET)
ARTICLE
|
doi:10.20944/preprints202406.0459.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
Protein kinase R, poxviruses, K3L, yatapoxvirus, translational regulation
Online: 7 June 2024 (08:08:13 CEST)
REVIEW
|
doi:10.20944/preprints201912.0412.v2
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Frank-Starling; angiotensin receptor; muscle contraction; myosin light chain kinase; Protein Kinase C-βII; myosin light chain phosphatase; β-arrestin; MgATP; MgADP-phosphomyosin; myosin LC affinity for Ca2+
Online: 11 January 2020 (13:24:08 CET)
REVIEW
|
doi:10.20944/preprints202107.0551.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
epidermal growth factor receptor; ErbB; biomarker; meningioma; intracranial tumor
Online: 23 July 2021 (22:06:24 CEST)
REVIEW
|
doi:10.20944/preprints202402.0872.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Immunotherapy; Immune checkpoint inhibitors; Rechallenge therapy; Resistance; NSCLC
Online: 16 February 2024 (11:34:11 CET)
ARTICLE
|
doi:10.20944/preprints202404.1231.v1
Subject:
Medicine And Pharmacology,
Pulmonary And Respiratory Medicine
Keywords:
apoptosis; diaphragm fibrosis; phosphoinositide 3-kinase-g; ventilator-induced diaphragm dysfunction
Online: 18 April 2024 (10:06:43 CEST)
REVIEW
|
doi:10.20944/preprints202406.0880.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Dendritic cells; DC based cancer vaccine; Immune checkpoint inhibitors; Cancer Therapy; Combinatorial therapy
Online: 13 June 2024 (11:51:42 CEST)
REVIEW
|
doi:10.20944/preprints202408.0744.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
Peripheral T-cell lymphoma; Histone deacetylase (HDAC); HDAC inhibitor (HDACi); targeted therapy; epigenetic; DNA mutation; TET2; DNMT3A
Online: 12 August 2024 (05:07:04 CEST)
ARTICLE
Subject:
Biology And Life Sciences,
Virology
Keywords:
JC virus; polyomavirus; SV40; progressive multifocal leukoencephalopathy
Online: 20 September 2020 (14:08:01 CEST)
ARTICLE
|
doi:10.20944/preprints202403.0717.v1
Subject:
Biology And Life Sciences,
Animal Science, Veterinary Science And Zoology
Keywords:
Lumpy skin disease; DNA polymerase; potential inhibitors; phytocompounds; antiviral drug compounds; molecular docking
Online: 13 March 2024 (07:58:39 CET)
REVIEW
|
doi:10.20944/preprints202408.1378.v1
Online: 19 August 2024 (16:27:50 CEST)
REVIEW
|
doi:10.20944/preprints202405.0832.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
multiple myeloma (MM); DNA damage response (DDR); mitogen‑activated protein kinase (MAPK); DDR-MAPK interplay; combination therapy
Online: 13 May 2024 (10:45:06 CEST)
REVIEW
|
doi:10.20944/preprints202205.0290.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
Cholesterol; PCSK9 inhibitors; HMG-CoA; LDL receptor; statins
Online: 23 May 2022 (10:01:24 CEST)
REVIEW
|
doi:10.20944/preprints202404.0091.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
menin; menin inhibitors; leukemia; KMT2A; NPM1
Online: 2 April 2024 (02:51:43 CEST)
ARTICLE
|
doi:10.20944/preprints202404.0426.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
CDK8; Cyclin C; Protein-protein interaction; Molecular dynamic simulation; Free energy calculation; Drug design
Online: 5 April 2024 (10:12:16 CEST)
ARTICLE
|
doi:10.20944/preprints202404.1491.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
HIV-2; integrase strand transfer inhibitor (INSTIs); HIV; integrase; Lenacapavir; SARs-CoV-2
Online: 23 April 2024 (05:06:50 CEST)
ARTICLE
|
doi:10.20944/preprints202407.0477.v1
Subject:
Medicine And Pharmacology,
Epidemiology And Infectious Diseases
Keywords:
DENV3; ZIKV; molecular docking; MD simulations; MM/GBSA; compound library; NS5; lycorine
Online: 5 July 2024 (12:04:10 CEST)
REVIEW
|
doi:10.20944/preprints202311.1503.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
receptor-type protein tyrosine phosphatases (RPTPs); CD148; R3 subgroup; Extracellular domain (ECD); Fibronectin; Polymorphisms; AlphaFold
Online: 23 November 2023 (10:53:39 CET)
ARTICLE
|
doi:10.20944/preprints202407.1450.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Bladder cancer; STAT3 inhibitor; Apoptosis; Preclinical; 3D models
Online: 17 July 2024 (14:18:54 CEST)
REVIEW
|
doi:10.20944/preprints202309.0682.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
Akt; cancer; metastasis; HNSCC; EMT; cytoskeletal remodelling
Online: 12 September 2023 (08:33:01 CEST)
ARTICLE
|
doi:10.20944/preprints202406.2011.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
machine learning; prediction methods; cancer; ic50; r programming
Online: 29 June 2024 (05:59:44 CEST)
ARTICLE
|
doi:10.20944/preprints202402.1740.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Rheumatoid Arthritis, Anti-TNF, NRF2, Reverse Signaling, Biotherapy, Monoclonal Antibodies, Monocytes, Prediction.
Online: 29 February 2024 (14:46:26 CET)
REVIEW
|
doi:10.20944/preprints202402.1049.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
malignant pleural mesothelioma; immune checkpoint inhibitor; orphan drug; good clinical practice; Pharmaceuticals and Medical Devices Agency
Online: 20 February 2024 (04:03:22 CET)
ARTICLE
|
doi:10.20944/preprints202405.1741.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
Alzheimer’ s disease; vascular complications; monoclonal antibody therapy; Aducanumab; Lecanemab; epoxide of polyunsaturated fatty acid; soluble epoxide hydrolase inhibitor EC5026; EP4 inhibitor; monocyte/macrophage; amyloid-beta degradation
Online: 27 May 2024 (13:00:54 CEST)
BRIEF REPORT
|
doi:10.20944/preprints202403.0928.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
systemic sclerosis; pulmonary hypertension; Phosphodiesterase-5 inhibitors; endothelin receptor antagonist
Online: 15 March 2024 (13:15:50 CET)
ARTICLE
|
doi:10.20944/preprints201906.0155.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
carboplatin; CIPN; TRPA1; cAMP; PKA; AKAP
Online: 17 June 2019 (09:53:39 CEST)
REVIEW
|
doi:10.20944/preprints202405.0573.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
Proton Pump Inhibitors (PPIs); Vonoprazan (VPZ); Intravenous infusion; Oral therapy; Bleeding peptic ulcers; Endoscopic therapy
Online: 9 May 2024 (09:15:54 CEST)
REVIEW
|
doi:10.20944/preprints202401.0310.v1
Subject:
Medicine And Pharmacology,
Dentistry And Oral Surgery
Keywords:
inflammation; inflammasome; inhibitors of the inflammasome; nanomaterials; functionalized biomaterials; periodontitis; general pathology
Online: 4 January 2024 (09:25:17 CET)
REVIEW
|
doi:10.20944/preprints202306.0441.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
anti-lipoxygenase peptide; bioactivity; enzymatic hydrolysis; food peptide; food protein; inflammation; lipoxidase; lipoxygenase inhibitory activity.
Online: 6 June 2023 (10:11:09 CEST)
ARTICLE
|
doi:10.20944/preprints202405.0035.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Mycobacterial Polyketide Synthase; QSAR; Multiple Linear Regression; Docking; Molecular Dynamics Simulations
Online: 1 May 2024 (16:46:55 CEST)
TECHNICAL NOTE
|
doi:10.20944/preprints202012.0641.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Neurodegeneration; dopamine; L-DOPA; dopaminergic; DBA; Western; IR; TH; Parkinson disease
Online: 25 December 2020 (07:10:33 CET)
ARTICLE
|
doi:10.20944/preprints201609.0123.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
carbonic anhydrase; acetylcholinesterase; β-Lactam; 2-Azetidinone; enzyme inhibition; enzyme purification
Online: 30 September 2016 (05:38:45 CEST)
ARTICLE
|
doi:10.20944/preprints202407.1916.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
cardiovascular disease; hepatic fibrosis; metabolic dysfunction-associated steatotic liver disease; sodium-glucose cotransporter 2 inhibitors; serum lipids
Online: 24 July 2024 (08:27:35 CEST)
ARTICLE
|
doi:10.20944/preprints202404.1152.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Tuberculosis; nitrobenzamides; DprE; mycobacteria
Online: 17 April 2024 (11:50:50 CEST)
ARTICLE
|
doi:10.20944/preprints202312.0533.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Colon tumorigenesis; ERK1/2; SOD3; migration, invasion; proliferation
Online: 8 December 2023 (04:56:53 CET)
REVIEW
|
doi:10.20944/preprints201807.0237.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
TRPM7, kinase, inflammation, lymphocytes, calcium signalling, SMAD, TH17, hypersensitivity, regulatory T cells, thrombosis, graft versus host disease, T cells, innate immunity
Online: 13 July 2018 (14:14:56 CEST)
REVIEW
|
doi:10.20944/preprints202204.0202.v1
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
Metabolic syndrome; SGLT2 inhibitors; Dapagliflozin; Empagliflozin; Canagliflozin; Translational modeling
Online: 21 April 2022 (10:12:04 CEST)
REVIEW
|
doi:10.20944/preprints202012.0167.v2
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Matrix metalloproteinase; MMPs; protease; TIMPs; exosite; small molecule inhibitors; monoclonal antibodies; proteomics; N-terminomics; TAILS
Online: 24 March 2021 (16:23:28 CET)
ARTICLE
|
doi:10.20944/preprints202406.0032.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
HIV-1; reverse transcriptase; polymerase; ribonuclease H; inhibitor; benzisothiazolone
Online: 3 June 2024 (07:56:06 CEST)
ARTICLE
|
doi:10.20944/preprints202306.1571.v1
Subject:
Chemistry And Materials Science,
Materials Science And Technology
Keywords:
cyclo-dipeptide; electrospinning; piezoelectricity; nanofibers; optical second harmonic generation; self-assembly
Online: 21 June 2023 (15:20:07 CEST)
REVIEW
|
doi:10.20944/preprints202401.0803.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
CYP enzymes; CYP3A4; flavonoid; inhibition; natural products
Online: 10 January 2024 (10:24:39 CET)
ARTICLE
|
doi:10.20944/preprints202307.0031.v1
Subject:
Chemistry And Materials Science,
Applied Chemistry
Keywords:
Ionic Liquids; Corrosion Inhibitors; Bio-based
Online: 4 July 2023 (02:23:59 CEST)
ARTICLE
|
doi:10.20944/preprints201710.0143.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
cheminformatics; docking simulation; drug repositioning; thiopurine; tyrosinase
Online: 22 October 2017 (14:03:13 CEST)
REVIEW
|
doi:10.20944/preprints202308.0709.v2
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
TLKs; DNA repair; HRR; NHEJ; replication; DNA damage; therapeutics
Online: 30 August 2023 (05:08:39 CEST)
ARTICLE
|
doi:10.20944/preprints202308.1008.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
diabetic vascular disease; endothelial cells; soluble vascular cell adhesion molecule 1
Online: 14 August 2023 (10:25:52 CEST)
ARTICLE
|
doi:10.20944/preprints202105.0297.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Protein Kinase Receptor (PKR); Mammarenavirus; Interferon; Innate immune response; Mx1; ISG15; CCL5
Online: 13 May 2021 (13:27:07 CEST)
REVIEW
|
doi:10.20944/preprints201809.0360.v1
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
p-21 activated kinase; pioglitazone, metformin, type 2 diabetes mellitus, cancer, chemoprevention, and inflammation.
Online: 19 September 2018 (00:50:05 CEST)
REVIEW
|
doi:10.20944/preprints201808.0403.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
p-21 activated kinase; pioglitazone, metformin, type 2 diabetes mellitus, cancer, chemoprevention, and inflammation.
Online: 23 August 2018 (05:10:55 CEST)
ARTICLE
|
doi:10.20944/preprints202403.1760.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
JAK-inhibitor; baricitinib; rheumatoid arthritis; real-word data; persistence; adherence; safety; unmet needs.
Online: 28 March 2024 (10:30:28 CET)
ARTICLE
|
doi:10.20944/preprints202208.0103.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Resveratrol; antioxidant metabolism; scavengome; biomimetic oxidation; bioactivity-guided isolation; NMR spectroscopy; xanthine oxidase
Online: 4 August 2022 (05:33:52 CEST)
ARTICLE
|
doi:10.20944/preprints202307.1689.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
N-acetyl-L-glutamate kinase; arginine biosynthesis; PII- signal transduction protein; green algae
Online: 25 July 2023 (11:43:42 CEST)
ARTICLE
|
doi:10.20944/preprints201807.0131.v1
Subject:
Medicine And Pharmacology,
Ophthalmology
Keywords:
pigmentary glaucoma; ROCK kinase inhibitor; RKI-1447; trabecular meshwork; phagocytosis; cytoskeleton
Online: 9 July 2018 (11:27:28 CEST)
ARTICLE
|
doi:10.20944/preprints201802.0026.v1
Subject:
Medicine And Pharmacology,
Ophthalmology
Keywords:
pig eye perfusion model; pigmentary glaucoma; ocular hypertension; ocular hypotension; phagocytosis; rho-kinase inhibitor
Online: 5 February 2018 (03:39:57 CET)
ARTICLE
|
doi:10.20944/preprints202310.1571.v2
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Transketolase; malonylation; acetylation; sirtuin 5; oxythiamine; metformin; amprolium; thiamine; posttranslational modifications
Online: 10 November 2023 (12:03:31 CET)
REVIEW
|
doi:10.20944/preprints202406.0356.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
liver transplantation; hepatocellular carcinoma; Immune checkpoint inhibitors; allograft rejection
Online: 6 June 2024 (07:45:00 CEST)
REVIEW
|
doi:10.20944/preprints202012.0419.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
immune checkpoint; lymphoid neoplasms; programmed death 1; cytotoxic T-lymphocyte antigen 4; monoclonal antibodies; combination therapies
Online: 17 December 2020 (08:10:05 CET)
CASE REPORT
|
doi:10.20944/preprints202406.1544.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
CFS (chronic fatigue syndrome), POTS (postural orthostatic tachycardia syndrome), stress, (COMT) catechol-O-methyltransferase, adrenaline, inflammation, AMPT (alpha-methyl-p-tyrosine)
Online: 21 June 2024 (14:43:51 CEST)
REVIEW
|
doi:10.20944/preprints202401.0297.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
dual leucine zipper kinase; phosphorylation; protein-protein interaction; proteasomal degradation; palmitoylation
Online: 4 January 2024 (09:32:03 CET)
REVIEW
|
doi:10.20944/preprints202309.1526.v1
Subject:
Biology And Life Sciences,
Neuroscience And Neurology
Keywords:
neurodegeneration with brain iron accumulation (NBIA); pantothenate kinaseassociated neurodegeneration (PKAN); pantothenate kinase 2 (PANK2); pantothenate; pantethine; vitamin E; omega 3; -lipoic acid; L-carnitine; thiamine; fibroblasts; induced neurons; precision medicine
Online: 22 September 2023 (09:18:39 CEST)
ARTICLE
|
doi:10.20944/preprints202305.0896.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
retinitis pigmentosa; cell death,; phosphoproteomic
Online: 12 May 2023 (07:17:25 CEST)
ARTICLE
|
doi:10.20944/preprints202205.0393.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
poxviruses; protein kinase R; evolution; translational regulation; eIF2
Online: 30 May 2022 (10:42:41 CEST)
ARTICLE
|
doi:10.20944/preprints202108.0100.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
PF-543; ceramide; SPHK; SPT; ceramide synthases; sphingolipid; metabolism; LC-MS/MS.
Online: 4 August 2021 (08:32:59 CEST)